SCHEMBL9623802

SCHEMBL9623802

CN(CCCc1ccc[n+]([O-])c1)CCCN1Cc2cc3c(cc2C1=O)OCO3

nearest known ligand 0.45

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GPR84 Q9NQS5 3/20 0.34
CYP2D6 P10635 2/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
ALDH1A1 P00352 1/20 0.32
GAA P10253 1/20 0.32
MAPK1 P28482 1/20 0.32
MAPK10 P53779 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9624289 0.91 CYP2D6 (0.37) GPR84CYP2D6CYP3A4KMT2A
SCHEMBL9624352 0.84 HCN4 (0.44) GPR84CYP3A4
SCHEMBL9624625 0.82 ALDH1A1 (0.41) ALDH1A1GAAMAPK1KMT2A
SCHEMBL9624482 0.82 TDP1 (0.34) CYP2D6
SCHEMBL9623778 0.81 EDNRB (0.36) CYP2D6CYP3A4ALDH1A1GAAMAPK1
SCHEMBL9624809 0.80 RAB9A (0.34) CYP2D6
SCHEMBL9625241 0.79 ALDH1A1 (0.36) CYP2D6CYP1A2CYP3A4ALDH1A1MAPK1
SCHEMBL9624353 0.79 SMN1; SMN2 (0.39)
SCHEMBL9623839 0.79 ALDH1A1 (0.41) ALDH1A1GAAMAPK1KMT2A
SCHEMBL9624157 0.77 MAPT (0.39) GPR84CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5116986-A HETEROAROMATIC AMINE DERIVATIVES DR. KARL THOMAE GMBH (DE) 1992-05-26 US disclosed
US-4912115-A Cardiovascular disorders DR. KARL THOMAE GMBH (DE) 1990-03-27 US disclosed