SCHEMBL9624482

SCHEMBL9624482

CN(CCCc1ccncc1)CCCN1Cc2cc3c(cc2C1=O)OCO3

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.34
PDE4A P27815 1/20 0.34
PDE4B Q07343 1/20 0.34
PDE4C Q08493 1/20 0.34
PDE4D Q08499 1/20 0.34
ALOX15 P16050 1/20 0.33
MAPT P10636 1/20 0.33
HCN4 Q9Y3Q4 1/20 0.33
CYP2D6 P10635 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9624380 0.90 MAPT (0.39) TDP1ALOX15MAPTHCN4CYP2D6
Hydrochloric Acid SCHEMBL9624724 0.89 CYP3A4 (0.40) ALOX15MAPTHCN4CYP2D6
SCHEMBL9624625 0.88 ALDH1A1 (0.41) TDP1ALOX15MAPT
SCHEMBL9624248 0.85 HDAC6 (0.35) ALOX15MAPTHCN4
SCHEMBL9623778 0.85 EDNRB (0.36) ALOX15MAPTHCN4CYP2D6
SCHEMBL9623839 0.84 ALDH1A1 (0.41) TDP1ALOX15MAPT
SCHEMBL9624809 0.84 RAB9A (0.34) MAPTHCN4CYP2D6
SCHEMBL9624353 0.83 SMN1; SMN2 (0.39)
SCHEMBL9624772 0.82 HCN4 (0.48) PDE4DALOX15MAPTHCN4
SCHEMBL9623802 0.82 GPR84 (0.34) CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5116986-A HETEROAROMATIC AMINE DERIVATIVES DR. KARL THOMAE GMBH (DE) 1992-05-26 US disclosed
US-4912115-A Cardiovascular disorders DR. KARL THOMAE GMBH (DE) 1990-03-27 US disclosed