SCHEMBL9623908

SCHEMBL9623908

CN(CCCN1Cc2cc3c(cc2C1=O)OCO3)CCc1ccc(Br)s1

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
MAPT P10636 1/20 0.32
HCN4 Q9Y3Q4 1/20 0.32
CYP2D6 P10635 1/20 0.32
SCN1A P35498 1/20 0.32
SCN2A Q99250 1/20 0.32
SCN3A Q9NY46 1/20 0.32
KDM4E B2RXH2 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
CYP3A4 P08684 1/20 0.32
ALOX15 P16050 1/20 0.32
SMPD1 P17405 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9624906 0.89 MAPT (0.32) KMT2AMAPTHCN4CYP2D6SCN1A
SCHEMBL9624678 0.87 HDAC6 (0.36) MAPTHCN4KDM4ETDP1CYP3A4
SCHEMBL9624293 0.84 HCN4 (0.46) MEN1KMT2AMAPTHCN4CYP3A4
SCHEMBL9624619 0.83 SMN1; SMN2 (0.37) SMN1; SMN2
SCHEMBL9624347 0.82 DRD2 (0.38)
SCHEMBL9624420 0.81 ALDH1A1 (0.36) SMN1; SMN2MAPTCYP2D6KDM4ECYP3A4
SCHEMBL9624911 0.81 MAPT (0.32) MEN1KMT2AMAPTHCN4CYP2D6
SCHEMBL9625345 0.81 CYP2D6 (0.32) MAPTHCN4CYP2D6SCN1ASCN2A
SCHEMBL9625096 0.80 MAPT (0.36) MAPTHCN4CYP3A4ALOX15SMPD1
SCHEMBL9625104 0.79 EDNRB (0.35) KMT2AMAPTHCN4CYP2D6SCN1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5116986-A HETEROAROMATIC AMINE DERIVATIVES DR. KARL THOMAE GMBH (DE) 1992-05-26 US disclosed
US-4912115-A Cardiovascular disorders DR. KARL THOMAE GMBH (DE) 1990-03-27 US disclosed
EP-0269968-A2 Heteroaromatic amine derivatives, medicaments containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1988-06-08 EP disclosed