SCHEMBL9624201

SCHEMBL9624201

Cc1cc2c(cc1C)C(=O)N(CCCN(C)CCc1cccnc1)C2

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 1/20 0.42
DHPS P49366 1/20 0.37
MAPT P10636 1/20 0.37
HCN4 Q9Y3Q4 1/20 0.37
SMPD1 P17405 1/20 0.36
CYP3A4 P08684 1/20 0.36
ALOX15 P16050 1/20 0.36
OPRM1 P35372 1/20 0.36
OPRL1 P41146 1/20 0.36
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
CRHR1 P34998 1/20 0.35
KCNA5 P22460 1/20 0.35
KCNJ5 P48544 1/20 0.35
KCNJ3 P48549 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10644226 0.96 CHRNA7 (0.40) CHRNA7DHPSOPRM1OPRL1KDM4E
SCHEMBL9625065 0.91 CHRNB2 (0.43) DHPSKDM4EALDH1A1
SCHEMBL9625087 0.90 MAPT (0.43) CHRNA7DHPSMAPTHCN4CYP3A4
SCHEMBL9624907 0.87 MAPT (0.49) CHRNA7MAPTHCN4SMPD1CYP3A4
SCHEMBL9623839 0.86 ALDH1A1 (0.41) CHRNA7MAPTALOX15OPRM1OPRL1
SCHEMBL9624387 0.86 MAPT (0.39) CHRNA7DHPSMAPTHCN4CYP3A4
SCHEMBL9624753 0.83 MAPT (0.45) MAPTHCN4CYP3A4ALOX15KDM4E
SCHEMBL9624248 0.83 HDAC6 (0.35) MAPTHCN4SMPD1CYP3A4ALOX15
SCHEMBL9624625 0.82 ALDH1A1 (0.41) CHRNA7MAPTALOX15OPRM1OPRL1
Hydrochloric Acid SCHEMBL9624866 0.82 CYP3A4 (0.46) MAPTHCN4CYP3A4ALOX15KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5116986-A HETEROAROMATIC AMINE DERIVATIVES DR. KARL THOMAE GMBH (DE) 1992-05-26 US disclosed
US-4912115-A Cardiovascular disorders DR. KARL THOMAE GMBH (DE) 1990-03-27 US disclosed
EP-0269968-A2 Heteroaromatic amine derivatives, medicaments containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1988-06-08 EP disclosed