SCHEMBL9624544

SCHEMBL9624544

Cc1cc2c(cc1C)CN(CCCN(C)CCc1ccsc1)C2

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 15/20 0.43
DRD2 P14416 2/20 0.40
DRD3 P35462 2/20 0.40
TP53 P04637 2/20 0.34
CYP1A2 P05177 2/20 0.34
CYP2D6 P10635 2/20 0.34
TSHR P16473 2/20 0.34
LTA4H P09960 1/20 0.34
GRIN2D O15399 1/20 0.33
GRIN3B O60391 1/20 0.33
CYP3A4 P08684 1/20 0.33
GRIN1 Q05586 1/20 0.33
GRIN2A Q12879 1/20 0.33
GRIN2B Q13224 1/20 0.33
GRIN2C Q14957 1/20 0.33
GRIN3A Q8TCU5 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9625041 0.87 SMPD1 (0.45) SIGMAR1CYP1A2CYP2D6CYP3A4
SCHEMBL9623557 0.86 SIGMAR1 (0.40) SIGMAR1DRD2DRD3
SCHEMBL9624476 0.81 MAPT (0.38) SIGMAR1DRD2DRD3LTA4HCYP3A4
SCHEMBL9625873 0.81 SMPD1 (0.35) SIGMAR1DRD2DRD3LTA4HCYP3A4
SCHEMBL9624612 0.78 LMNA (0.46) SIGMAR1TSHR
SCHEMBL9623887 0.76 HDAC6 (0.34) DRD2DRD3LTA4HCYP3A4
SCHEMBL9624635 0.76 CHRNA7 (0.49) SIGMAR1
SCHEMBL9624963 0.75 HDAC6 (0.34) SIGMAR1DRD2DRD3LTA4HCYP3A4
SCHEMBL9624528 0.75 LMNA (0.46) SIGMAR1DRD3TSHR
SCHEMBL9625068 0.74 HDAC6 (0.35) SIGMAR1DRD2DRD3LTA4HCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5116986-A HETEROAROMATIC AMINE DERIVATIVES DR. KARL THOMAE GMBH (DE) 1992-05-26 US disclosed
US-4912115-A Cardiovascular disorders DR. KARL THOMAE GMBH (DE) 1990-03-27 US disclosed