SCHEMBL9624867

SCHEMBL9624867

CC/C=C(\CCC)C(=O)Cl

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.46
CES2 O00748 1/20 0.38
CES1 P23141 1/20 0.38
ALDH1A1 P00352 3/20 0.37
TP53 P04637 1/20 0.37
HDAC3 O15379 4/20 0.36
HDAC1 Q13547 4/20 0.36
HDAC2 Q92769 4/20 0.36
HDAC8 Q9BY41 4/20 0.36
FFAR3 O14843 3/20 0.36
GRIK1 P39086 1/20 0.35
GRIK2 Q13002 1/20 0.35
HDAC6 Q9UBN7 1/20 0.32
TDP1 Q9NUW8 1/20 0.31
CTSD P07339 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22268157 0.80
SCHEMBL9493661 0.78 GRIK1 (0.50) TSHRCES2CES1ALDH1A1HDAC3
SCHEMBL691600 0.78 GRIK1 (0.50) TSHRCES2CES1ALDH1A1HDAC3
SCHEMBL25932051 0.78 CES1 (0.52) TSHRCES2CES1ALDH1A1HDAC3
SCHEMBL11243324 0.78 CES1 (0.39) TSHRCES2CES1ALDH1A1HDAC3
SCHEMBL1003142 0.78 GRIK1 (0.50) TSHRCES2CES1ALDH1A1HDAC3
SCHEMBL11243321 0.78 CES1 (0.39) TSHRCES2CES1ALDH1A1HDAC3
SCHEMBL11288817 0.76 GRIK1 (0.39) TSHRCES2CES1ALDH1A1TP53
SCHEMBL11288814 0.76 GRIK1 (0.39) TSHRCES2CES1ALDH1A1TP53
Hydrochloric Acid SCHEMBL9624870 0.76 GRIK1 (0.48) TSHRCES2CES1ALDH1A1HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5162573-A Anticonvulsant, antiepileptic agent CHIESI FARMACEUTICI S.P.A. (IT) 1992-11-10 US disclosed
EP-0250997-B1 VALPROIC AND (E)-2-VALPROENOIC ACID DERIVATIVES, PROCESSES FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS THEREFROM CHIESI FARMACEUTICI S.p.A. (IT) 1992-04-15 EP disclosed
EP-0250997-A2 Valproic and (E)-2-valproenoic acid derivatives, processes for the preparation thereof and pharmaceutical compositions therefrom CHIESI FARMACEUTICI S.p.A. (IT) 1988-01-07 EP disclosed