SCHEMBL9624873

SCHEMBL9624873

Cc1ccc(CCN(C)CCCN2Cc3cc(C)c(C)cc3C2=O)s1

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 1/20 0.35
MAPT P10636 2/20 0.34
HCN4 Q9Y3Q4 1/20 0.34
CYP3A4 P08684 1/20 0.34
ALOX15 P16050 1/20 0.34
KDM4E B2RXH2 2/20 0.33
ALDH1A1 P00352 2/20 0.33
HPGD P15428 2/20 0.33
SMPD1 P17405 1/20 0.32
PRF1 P14222 1/20 0.31
MEN1 O00255 1/20 0.31
GAA P10253 1/20 0.31
THRB P10828 1/20 0.31
KMT2A Q03164 1/20 0.31
HSD17B10 Q99714 1/20 0.31
DRD2 P14416 1/20 0.30
DRD3 P35462 1/20 0.30
KCNH2 Q12809 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9624678 0.89 HDAC6 (0.36) HDAC6MAPTHCN4CYP3A4ALOX15
SCHEMBL9624752 0.88 HCN4 (0.46) MAPTHCN4CYP3A4ALOX15KDM4E
SCHEMBL9624906 0.88 MAPT (0.32) MAPTHCN4CYP3A4ALOX15KMT2A
SCHEMBL9625527 0.84 L3MBTL1 (0.38) HDAC6MAPTHCN4ALDH1A1SMPD1
SCHEMBL9624431 0.83 HDAC6 (0.33) HDAC6MAPTHCN4CYP3A4ALOX15
SCHEMBL9625705 0.83 DRD2 (0.39) HDAC6SMPD1DRD2DRD3KCNH2
SCHEMBL9624575 0.80 CES2 (0.35) HDAC6MAPTHCN4CYP3A4ALOX15
SCHEMBL9624134 0.80 L3MBTL1 (0.38) HDAC6ALDH1A1MEN1KMT2ADRD3
SCHEMBL9624774 0.80 HDAC6 (0.36) HDAC6MAPTHCN4CYP3A4ALOX15
SCHEMBL9624476 0.80 MAPT (0.38) HDAC6MAPTHCN4CYP3A4ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5116986-A HETEROAROMATIC AMINE DERIVATIVES DR. KARL THOMAE GMBH (DE) 1992-05-26 US disclosed
US-4912115-A Cardiovascular disorders DR. KARL THOMAE GMBH (DE) 1990-03-27 US disclosed
EP-0269968-A2 Heteroaromatic amine derivatives, medicaments containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1988-06-08 EP disclosed