SCHEMBL9624904

SCHEMBL9624904

CN(CCCN1CCc2c(ccc3c2OCO3)C1=O)CCc1ccsc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.37
HCN4 Q9Y3Q4 1/20 0.37
CYP3A4 P08684 2/20 0.36
ALOX15 P16050 1/20 0.36
KDM4E B2RXH2 2/20 0.33
CYP2D6 P10635 2/20 0.33
CYP2C19 P33261 2/20 0.33
TSHR P16473 1/20 0.33
SIGMAR1 Q99720 3/20 0.32
CTSL P07711 1/20 0.32
NAAA Q02083 1/20 0.32
BCHE P06276 2/20 0.31
SMPD1 P17405 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
LTA4H P09960 1/20 0.30
MAOA P21397 1/20 0.30
ACHE P22303 1/20 0.30
MAOB P27338 1/20 0.30
DRD2 P14416 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10401291 0.95 NAAA (0.36) MAPTHCN4CYP3A4ALOX15KDM4E
SCHEMBL9625000 0.87 CNR2 (0.39) MAPTHCN4CYP3A4ALOX15KDM4E
SCHEMBL9624670 0.85 CYP3A4 (0.34) MAPTHCN4CYP3A4ALOX15KDM4E
SCHEMBL9624078 0.82 MAPT (0.39) MAPTHCN4CYP3A4ALOX15KDM4E
SCHEMBL9624416 0.81 KDM4E (0.34) MAPTHCN4CYP3A4ALOX15KDM4E
SCHEMBL9624338 0.81 SIGMAR1 (0.34) MAPTHCN4CYP3A4ALOX15KDM4E
SCHEMBL9624644 0.79 DRD2 (0.33) MAPTHCN4CYP3A4ALOX15KDM4E
SCHEMBL9624412 0.79 KDM4E (0.34) MAPTHCN4CYP3A4ALOX15KDM4E
SCHEMBL9625002 0.79 DRD2 (0.33) MAPTHCN4CYP3A4ALOX15KDM4E
SCHEMBL9625302 0.79 MAPT (0.36) MAPTHCN4CYP3A4ALOX15KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5116986-A HETEROAROMATIC AMINE DERIVATIVES DR. KARL THOMAE GMBH (DE) 1992-05-26 US disclosed
US-4912115-A Cardiovascular disorders DR. KARL THOMAE GMBH (DE) 1990-03-27 US disclosed