SCHEMBL9625629

SCHEMBL9625629

CN(C)c1ccc2[c]csc2c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.37
TSHR P16473 4/20 0.37
ALOX15 P16050 3/20 0.37
HSD17B10 Q99714 2/20 0.37
APP P05067 5/20 0.35
TERT O14746 1/20 0.35
MAPT P10636 4/20 0.33
INSR P06213 1/20 0.33
MAPK1 P28482 5/20 0.32
TDP1 Q9NUW8 5/20 0.32
SMN1; SMN2 Q16637 4/20 0.32
KDM4E B2RXH2 4/20 0.32
THRB P10828 3/20 0.32
RECQL P46063 3/20 0.32
MEN1 O00255 2/20 0.32
APAF1 O14727 2/20 0.32
GSR P00390 2/20 0.32
POLB P06746 2/20 0.32
PKM P14618 2/20 0.32
MAOA P21397 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9625533 0.80 TERT (0.41) ALDH1A1TSHRALOX15HSD17B10TERT
SCHEMBL207512 0.69 CYP2A6 (0.35)
SCHEMBL9624198 0.69 ALDH1A1 (0.35) ALDH1A1TSHRALOX15HSD17B10MAPT
SCHEMBL9624098 0.69 NOX1 (0.31)
SCHEMBL5538925 0.65 EPHX2 (0.39) ALDH1A1TSHRHSD17B10MAPK1KDM4E
SCHEMBL827260 0.64 APP (0.47) ALDH1A1TSHRALOX15HSD17B10APP
SCHEMBL16288692 0.63
SCHEMBL1147598 0.61 APP (0.39) ALDH1A1TSHRALOX15HSD17B10APP
SCHEMBL6357105 0.61 ALDH1A1 (0.37) ALDH1A1TSHRALOX15HSD17B10APP
SCHEMBL926598 0.61 TDP1 (0.47) ALDH1A1ALOX15HSD17B10APPTERT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5116986-A HETEROAROMATIC AMINE DERIVATIVES DR. KARL THOMAE GMBH (DE) 1992-05-26 US claimed
US-4912115-A Cardiovascular disorders DR. KARL THOMAE GMBH (DE) 1990-03-27 US claimed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed
US-5116986-A HETEROAROMATIC AMINE DERIVATIVES DR. KARL THOMAE GMBH (DE) 1992-05-26 US disclosed
US-4912115-A Cardiovascular disorders DR. KARL THOMAE GMBH (DE) 1990-03-27 US disclosed