SCHEMBL9628583

SCHEMBL9628583

CCCN(C)CC1CCc2ccc(O)cc21

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.55
ESR2 Q92731 1/20 0.55
DRD2 P14416 6/20 0.52
DRD3 P35462 6/20 0.52
DRD4 P21917 4/20 0.52
NQO2 P16083 1/20 0.51
MTNR1A P48039 1/20 0.51
MTNR1B P49286 1/20 0.51
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
OPRM1 P35372 2/20 0.50
OPRD1 P41143 2/20 0.50
OPRK1 P41145 2/20 0.50
CYP2D6 P10635 2/20 0.50
HTR1A P08908 1/20 0.50
ADRB2 P07550 1/20 0.50
CASP1 P29466 1/20 0.50
LMNA P02545 3/20 0.49
MAPT P10636 1/20 0.49
TSHR P16473 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9627819 0.89 ADRA2A (0.57) ESR1ESR2DRD2DRD3DRD4
SCHEMBL9628347 0.85 ESR1 (0.60) ESR1ESR2DRD2DRD3DRD4
SCHEMBL9629977 0.83 ESR1 (0.52) ESR1ESR2DRD2DRD3DRD4
SCHEMBL9628446 0.82 ESR1 (0.57) ESR1ESR2DRD2DRD3DRD4
SCHEMBL11652411 0.80 ESR1 (0.66) ESR1ESR2NQO2MTNR1AMTNR1B
SCHEMBL9629909 0.79 DRD2 (0.55) ESR1ESR2DRD2DRD3DRD4
SCHEMBL9627834 0.75 DRD3 (0.45) DRD2DRD3DRD4MEN1KMT2A
SCHEMBL9627796 0.74 NQO2 (0.57) ESR1ESR2DRD2DRD3DRD4
SCHEMBL9308578 0.73 DRD2 (0.66) DRD2DRD3DRD4MEN1KMT2A
SCHEMBL9308579 0.73 DRD2 (0.66) DRD2DRD3DRD4MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0281261-B1 3-AMINOMETHYL DERIVATIVES OF INDANE, INDOLINE AND DIHYDROBENZOFURANE AND DIHYDROBENZOTHIOPHENE H. LUNDBECK A/S (DK) 1992-05-06 EP disclosed
US-4946863-A CNS-affecting 6-oxy-3-aminomethyl indanes, compositions thereof, and method of treating therewith H. LUNDBECK A/S (DK) 1990-08-07 US disclosed
US-4847254-A CNS affecting 5-oxy-3-aminomethyl-dihydro-benzofurans and benzothiophenes H. LUNDBECK A/S (DK) 1989-07-11 US disclosed
EP-0281261-A2 3-Aminomethyl derivatives of indane, indoline and dihydrobenzofurane and dihydrobenzothiophene H. LUNDBECK A/S (DK) 1988-09-07 EP disclosed