SCHEMBL9628819

SCHEMBL9628819

CC(C)NC(Oc1ccc(C(C)C(=O)O)cc1)C(C)O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 9/20 0.44
AKR1C3 P42330 8/20 0.44
PTGS1 P23219 7/20 0.44
AKR1C2 P52895 7/20 0.44
TSHR P16473 2/20 0.44
SLC22A6 Q4U2R8 2/20 0.44
CDC42 P60953 1/20 0.44
RAC1 P63000 1/20 0.44
CYP1A2 P05177 1/20 0.44
LMNA P02545 2/20 0.41
CYP2C9 P11712 2/20 0.41
CXCR1 P25024 2/20 0.41
CXCR2 P25025 2/20 0.41
ALB P02768 1/20 0.41
ESR1 P03372 1/20 0.41
ALOX5 P09917 1/20 0.41
RARB P10826 1/20 0.41
ADRB3 P13945 1/20 0.41
NFKB1 P19838 1/20 0.41
HTR2A P28223 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10345923 0.79 LMNA (0.41) TSHRCYP1A2LMNACYP2C9ADRB3
SCHEMBL21775493 0.77 KMT2A (0.41) LMNAADRB3
SCHEMBL27579668 0.77 KMT2A (0.60) PTGS2AKR1C3PTGS1AKR1C2TSHR
SCHEMBL21775539 0.75 AOC3 (0.39) ADRB3CNR2
SCHEMBL10881708 0.74 PTGS2 (0.52) PTGS2AKR1C3PTGS1AKR1C2TSHR
SCHEMBL9484088 0.74 LMNA (0.53) TSHRCYP1A2LMNANFKB1BLM
SCHEMBL11392495 0.73 PABPC1 (0.35) ADRB3PMP22CNR2
SCHEMBL2585659 0.73 PPARG (0.39) CYP1A2LMNAADRB3CNR2CYP2C19
SCHEMBL28243247 0.72 PTGS2 (0.50) PTGS2AKR1C3PTGS1AKR1C2TSHR
SCHEMBL20552868 0.72 PPARG (0.43) TSHRCYP1A2LMNAADRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0256586-B1 PROCESS FOR THE PREPARATION OF ESTERS OF 4-(2,3-EPOXYPROPOXY)PHENYLACETIC ACID AND 4-(2-HYDROXY-3-ISOPROPYLAMINO-PROPOXY)PHENYLACETIC ACID AND/OR ATENOLOL IN STEREOSPECIFIC FORM GIST-BROCADES N.V. (NL) 1992-05-13 EP disclosed