SCHEMBL9629316

SCHEMBL9629316

Fc1ccc(CCN2CCCCC2)cc1

nearest known ligand 0.78

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 6/20 0.71
SIGMAR1 Q99720 2/20 0.66
L3MBTL1 Q9Y468 2/20 0.66
MBTD1 Q05BQ5 1/20 0.66
L3MBTL3 Q96JM7 1/20 0.66
SCN5A Q14524 1/20 0.64
SLC6A3 Q01959 2/20 0.62
CYP1A2 P05177 1/20 0.61
CYP3A4 P08684 1/20 0.61
MAOA P21397 1/20 0.59
KCNJ1 P48048 1/20 0.58
KCNH2 Q12809 1/20 0.58
TDP1 Q9NUW8 1/20 0.58
HTR2A P28223 1/20 0.54
HTR2C P28335 1/20 0.54
HTR7 P34969 1/20 0.54
HTR6 P50406 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23377646 0.98 HRH3 (0.68) HRH3SIGMAR1L3MBTL1MBTD1L3MBTL3
SCHEMBL23377845 0.94 HRH3 (0.62) HRH3SIGMAR1L3MBTL1MBTD1L3MBTL3
SCHEMBL6984190 0.89 SCN5A (0.74) HRH3SIGMAR1SCN5ASLC6A3HTR2A
SCHEMBL22813547 0.86 SCN5A (0.71) HRH3SIGMAR1SCN5ASLC6A3HTR2A
SCHEMBL5752571 0.83 KCNH2 (0.64) HRH3SIGMAR1L3MBTL1MBTD1L3MBTL3
SCHEMBL5745400 0.82 KCNJ1 (0.61) HRH3SIGMAR1SLC6A3CYP1A2MAOA
SCHEMBL8804098 0.82 MAOA (0.67) HRH3SIGMAR1L3MBTL1MBTD1L3MBTL3
SCHEMBL23731966 0.82 SCN5A (0.66) HRH3SIGMAR1SCN5ASLC6A3HTR2A
SCHEMBL13958507 0.82 L3MBTL1 (0.96) HRH3SIGMAR1L3MBTL1MBTD1L3MBTL3
SCHEMBL13958981 0.82 L3MBTL1 (0.96) HRH3SIGMAR1L3MBTL1MBTD1L3MBTL3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101412693-A 4-[1-hydroxy-1-(2,3-dimethoxyphenyl)methyl]piperidine and method for preparing corresponding piperidine thereby AVENTIS PHARMA INC (US) 2009-04-22 CN disclosed
CN-1989119-A New benzoyl urea derivatives RICHTER GEDEON VEGYESZET (HU) 2007-06-27 CN disclosed
CN-1143321-A Treatment of obsessive-compulsive disorders with 5-HT2 antagonists MERRELL DOW PHARMA (US) 1997-02-19 CN disclosed
US-5134149-A Serotonin antagonist MERRELL DOW PHARMACEUTICALS INC. (US) 1992-07-28 US disclosed