SCHEMBL9629472

SCHEMBL9629472

Nc1ccncc1NC(=S)NCCN1CCC(Nc2nc3cccnc3n2Cc2cccs2)C1

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 1/20 0.38
ROCK2 O75116 6/20 0.35
CCR2 P41597 5/20 0.35
ROCK1 Q13464 5/20 0.35
MAPT P10636 9/20 0.35
TP53 P04637 5/20 0.35
ENPP2 Q13822 1/20 0.34
POLB P06746 1/20 0.34
GAA P10253 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9630310 0.90 EED (0.40) ROCK2CCR2ROCK1MAPTTP53
SCHEMBL9631303 0.87 ROCK2 (0.35) ROCK2CCR2ROCK1TP53
SCHEMBL9629497 0.87 ROCK2 (0.34) ROCK2CCR2ROCK1MAPTTP53
SCHEMBL9691136 0.86 SLC6A9 (0.44) SLC6A9MAPTTP53ENPP2POLB
SCHEMBL10548020 0.85 SLC6A9 (0.53) SLC6A9MAPTTP53ENPP2POLB
SCHEMBL1152028 0.84 HRH1 (0.38) ROCK2CCR2ROCK1MAPTTP53
SCHEMBL1152449 0.83 KCNH2 (0.46) ROCK2CCR2ROCK1MAPTTP53
SCHEMBL9690741 0.82 SLC6A9 (0.46) SLC6A9MAPTTP53ENPP2POLB
SCHEMBL10382581 0.80 SLC6A9 (0.36) SLC6A9ROCK2ROCK1MAPTTP53
SCHEMBL9629312 0.80 SLC6A9 (0.47) SLC6A9ROCK2CCR2ROCK1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5151424-A Antiallergens or antihistamines JANSSEN PHARMACEUTICA N.V. (BE) 1992-09-29 US disclosed
US-5071846-A Anti-hystaminic [(bicyclic heterocyclyl) methyl and --hetero] substituted hexahydro-1H-azepines and pyrrolidines JANSSEN PHARMACEUTICA N.V. (BE) 1991-12-10 US disclosed
US-4988689-A Antiallergens, antihistamines JANSSEN PHARMACEUTICA N.V. (BE) 1991-01-29 US disclosed