SCHEMBL9629983

SCHEMBL9629983

O=c1c(N2CCCCC2)c(O)c2cccnc2n1-c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FEN1 P39748 1/20 0.51
ALDH1A1 P00352 3/20 0.48
KDM4E B2RXH2 2/20 0.48
PDE4A P27815 7/20 0.47
PDE4B Q07343 6/20 0.47
PDE4C Q08493 6/20 0.47
PDE4D Q08499 6/20 0.47
TSHR P16473 2/20 0.44
CYP2C19 P33261 2/20 0.44
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
LMNA P02545 1/20 0.43
PDE1A P54750 1/20 0.42
PDE1B Q01064 1/20 0.42
LOXL3 P58215 1/20 0.41
LOXL2 Q9Y4K0 1/20 0.41
GAA P10253 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Water SCHEMBL9629740 0.99 FEN1 (0.50) FEN1ALDH1A1KDM4EPDE4APDE4B
Pirodomast SCHEMBL125348 0.99 FEN1 (0.52) FEN1ALDH1A1KDM4EPDE4APDE4B
Pirodomast SCHEMBL29385413 0.99 FEN1 (0.52) FEN1ALDH1A1KDM4EPDE4APDE4B
Pirodomast SCHEMBL9488218 0.98 FEN1 (0.51) FEN1ALDH1A1KDM4EPDE4APDE4B
SCHEMBL9629745 0.87 FEN1 (0.48) FEN1ALDH1A1KDM4EPDE4APDE4B
Water SCHEMBL10427748 0.87 MAPT (0.44) FEN1ALDH1A1KDM4EPDE4BPDE4D
Water SCHEMBL9629016 0.86 FEN1 (0.47) FEN1ALDH1A1KDM4EPDE4APDE4B
Pirodomast SCHEMBL607268 0.86 LOXL3 (0.43) FEN1ALDH1A1KDM4EPDE4APDE4B
Water SCHEMBL10582943 0.84 FEN1 (0.46) FEN1ALDH1A1PDE4APDE4BPDE4C
Water SCHEMBL10580186 0.81 ALDH1A1 (0.43) FEN1ALDH1A1KDM4EPDE4APDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0232328-B1 ZWITTERIONIC BICYCLIC COMPOUNDS AND THEIR SALTS, SOLVATES, HYDRATES AND ESTERS SCHERING CORPORATION (US) 1992-04-15 EP claimed
EP-0338010-B1 PHARMACEUTICAL COMPOSITIONS FOR TREATMENT OF HYPERPROLIFERATE SKIN DISEASE SCHERING CORPORATION (US) 1992-02-05 EP claimed