SCHEMBL9632167

SCHEMBL9632167

CC(=O)Oc1c(C)c(C)c2c(c1C)C(=O)CC(COc1ccc(N)cc1)(CC(C)C)O2

nearest known ligand 0.34

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
PDE4A P27815 1/20 0.34
PDE3A Q14432 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9631440 0.88 KMT2A (0.38) MEN1KMT2APDE4APDE3A
SCHEMBL9631349 0.87 MEN1 (0.47) MEN1KMT2APDE4APDE3A
SCHEMBL9632620 0.85 MEN1 (0.33) MEN1KMT2APDE4APDE3A
SCHEMBL9632313 0.84 MEN1 (0.30) MEN1KMT2APDE4APDE3A
SCHEMBL7125937 0.84 MEN1 (0.36) MEN1KMT2APDE4APDE3A
SCHEMBL10641768 0.83 MEN1 (0.46) MEN1KMT2APDE4APDE3A
SCHEMBL9630744 0.76 MEN1 (0.46) MEN1KMT2APDE4APDE3A
SCHEMBL10640049 0.74 MEN1 (0.42) MEN1KMT2APDE4APDE3A
SCHEMBL9632039 0.74 NPC1 (0.36) MEN1KMT2A
SCHEMBL9631403 0.74 MEN1 (0.42) MEN1KMT2APDE4APDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5104888-A Anticholesterol or antidiabetic agents SANKYO COMPANY, LIMITED (JP) 1992-04-14 US disclosed
EP-0207581-B1 THIAZOLIDINE DERIVATIVES, THEIR PREPARATION AND USE SANKYO COMPANY LIMITED (JP) 1990-09-12 EP disclosed
EP-0207581-A2 Thiazolidine derivatives, their preparation and use SANKYO COMPANY LIMITED (JP) 1987-01-07 EP disclosed