SCHEMBL9632335

SCHEMBL9632335

N#Cc1ccc2c(c1F)C(=O)NC2=O

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 3/20 0.41
GRM5 P41594 4/20 0.39
PPOX P50336 1/20 0.36
EGLN2 Q96KS0 3/20 0.36
CHEK1 O14757 3/20 0.35
GSK3B P49841 1/20 0.34
UPP1 Q16831 1/20 0.34
PTP4A3 O75365 1/20 0.34
WEE1 P30291 2/20 0.33
AR P10275 1/20 0.33
ALK Q9UM73 1/20 0.32
USP8 P40818 1/20 0.32
USP7 Q93009 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11426926 0.80 PARP1 (0.42) PARP1GRM5PPOXCHEK1GSK3B
SCHEMBL29710128 0.77 GRM5 (0.46) PARP1GRM5PPOXCHEK1GSK3B
SCHEMBL9279015 0.77 GRM5 (0.46) PARP1GRM5PPOXCHEK1GSK3B
SCHEMBL28920768 0.75 GRM5 (0.44) PARP1GRM5PPOXCHEK1GSK3B
SCHEMBL9489040 0.74 GSK3B (0.46) PARP1CHEK1GSK3BWEE1USP8
SCHEMBL29704524 0.73 GSK3B (0.45) PARP1CHEK1GSK3BWEE1USP8
SCHEMBL28099608 0.69 PARP1 (0.46) PARP1GRM5PPOXCHEK1GSK3B
SCHEMBL6651902 0.68 TRPV4 (0.48) EGLN2UPP1AR
Phosphoric Acid SCHEMBL30230307 0.68 GRM5 (0.39) PARP1GRM5PPOXCHEK1GSK3B
SCHEMBL7943820 0.68 USP8 (0.47) GRM5PPOXCHEK1GSK3BUPP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0484381-A1 N-CYANOIMIDES AND PROCESS FOR THEIR PREPARATION AND USES THEREOF HENKEL RESEARCH CORPORATION (US) 1992-05-13 EP disclosed
WO-1991001307-A2 N-CYANOIMIDES AND PROCESS FOR THEIR PREPARATION AND USES THEREOF HENKEL RESEARCH CORPORATION (US) 1991-02-07 WO disclosed