SCHEMBL9633635

SCHEMBL9633635

COc1ccc(F)cc1OCC=O

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TUBB1 Q9H4B7 1/20 0.54
FFAR1 O14842 1/20 0.49
FFAR4 Q5NUL3 1/20 0.49
ALDH1A1 P00352 3/20 0.47
MEN1 O00255 1/20 0.47
POLB P06746 1/20 0.47
HPGD P15428 1/20 0.47
KMT2A Q03164 1/20 0.47
NFE2L2 Q16236 2/20 0.45
HTR1A P08908 3/20 0.42
CTSL P07711 2/20 0.42
CTSS P25774 2/20 0.42
CTSK P43235 2/20 0.42
KDM4E B2RXH2 1/20 0.42
TSHR P16473 1/20 0.42
PTGS1 P23219 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C19 P33261 1/20 0.41
ERN1 O75460 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9631899 0.87 TUBB1 (0.44) TUBB1FFAR1FFAR4ALDH1A1MEN1
SCHEMBL16741066 0.83 CTSS (0.46) TUBB1ALDH1A1MEN1POLBHPGD
SCHEMBL17848603 0.82 CTSS (0.42) TUBB1ALDH1A1MEN1POLBHPGD
SCHEMBL29863189 0.81 MRGPRX4 (0.47) TUBB1FFAR1FFAR4ALDH1A1MEN1
SCHEMBL18715363 0.81 ACHE (0.59) TUBB1ALDH1A1MEN1POLBHPGD
SCHEMBL20578753 0.80 POLB (0.50) TUBB1ALDH1A1MEN1POLBHPGD
SCHEMBL2555360 0.80 CTSS (0.53) ALDH1A1MEN1POLBHPGDKMT2A
SCHEMBL514581 0.80 CA1 (0.54) TUBB1POLBHTR1ACTSLCTSS
SCHEMBL16422054 0.79 MRGPRX1 (0.40) TUBB1ALDH1A1MEN1POLBKMT2A
Butanal SCHEMBL10751573 0.78 NFE2L2 (0.47) FFAR1FFAR4ALDH1A1MEN1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0331943-B1 PHENOXYETHYLAMINE DERIVATIVES, PROCESS FOR PREPARING THE SAME, AND COMPOSITION FOR EXHIBITING EXCELLENT ALPHA-1-BLOCKING ACTIVITY CONTAINING THE SAME Hokuriku Pharmaceutical Co.,Ltd (JP) 1992-06-17 EP disclosed
US-4971990-A HYPOTENSIVE AGENTS, DYSUREA HOKURIKU PHARMACEUTICAL CO., LTD. (JP) 1990-11-20 US disclosed
EP-0331943-A1 Phenoxyethylamine derivatives, process for preparing the same, and composition for exhibiting excellent alpha-1-blocking activity containing the same Hokuriku Pharmaceutical Co.,Ltd (JP) 1989-09-13 EP disclosed