SCHEMBL9633804

SCHEMBL9633804

COC(=O)c1ccc(Cc2cccc3ccc(C(N)=O)cc23)c(OC)c1

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NQO2 P16083 2/20 0.48
MTNR1A P48039 7/20 0.45
MAPT P10636 1/20 0.44
PLAU P00749 2/20 0.43
PLAT P00750 1/20 0.43
MAPK1 P28482 1/20 0.42
GPR84 Q9NQS5 1/20 0.41
PARP15 Q460N3 1/20 0.41
PARP10 Q53GL7 1/20 0.41
PLA2G4A P47712 1/20 0.41
CHEK2 O96017 1/20 0.40
MTNR1B P49286 1/20 0.40
TRPV1 Q8NER1 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9634717 0.90 PLA2G4A (0.51) MTNR1AMAPK1PLA2G4A
SCHEMBL9634970 0.90 NQO2 (0.49) NQO2MTNR1APLA2G4AMTNR1B
SCHEMBL9633886 0.89 MAPT (0.49) NQO2MTNR1AMAPTPLAUMAPK1
SCHEMBL9633776 0.84 NQO2 (0.44) NQO2MTNR1AMAPTMTNR1B
SCHEMBL9634228 0.84 PLA2G4A (0.51) NQO2MTNR1AMAPTPLAUPLA2G4A
SCHEMBL9634171 0.83 PLA2G4A (0.53) PLA2G4A
SCHEMBL9633803 0.83 NQO2 (0.48) NQO2
SCHEMBL9633708 0.81 NQO2 (0.47) NQO2
SCHEMBL9634320 0.81 CYP1A2 (0.50) NQO2MTNR1AMAPTMTNR1B
SCHEMBL9634206 0.81 NQO2 (0.46) NQO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0337765-B1 ACYLSULFONAMIDE DERIVATIVES OF ALPHA-CARBOCYCLYLTOLUIC ACIDS USED AS LEUKOTRIENE ANTAGONISTS ICI AMERICAS INC. (US) 1992-10-14 EP disclosed
US-5095038-A Antiinflammatory, antiallergens ICI AMERICAS INC. (US) 1992-03-10 US disclosed
EP-0337765-A2 Acylsulfonamide derivatives of alpha-carbocyclyltoluic acids used as leukotriene antagonists ICI AMERICAS INC. (US) 1989-10-18 EP disclosed