SCHEMBL9634320

SCHEMBL9634320

COC(=O)c1ccc(Cc2cccc3ccc(CCCC(=O)O)cc23)c(OC)c1

nearest known ligand 0.50

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2C19 P33261 1/20 0.50
MTNR1A P48039 7/20 0.45
MTNR1B P49286 4/20 0.45
NQO2 P16083 2/20 0.44
CYP4A11 Q02928 2/20 0.41
CYP4F2 P78329 1/20 0.41
TLR7 Q9NYK1 1/20 0.40
SELP P16109 1/20 0.40
MAPT P10636 1/20 0.39
ALDH1A1 P00352 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9633818 0.89 NQO2 (0.42) CYP1A2CYP2D6CYP2C19MTNR1AMTNR1B
SCHEMBL9633707 0.88 KMT2A (0.41) CYP1A2CYP2D6CYP2C19MTNR1AMTNR1B
SCHEMBL9634229 0.85 PPARA (0.43) MTNR1AMTNR1BNQO2MAPT
SCHEMBL9634970 0.84 NQO2 (0.49) MTNR1AMTNR1BNQO2
SCHEMBL9633717 0.84 KMT2A (0.46) MTNR1AMTNR1BNQO2ALDH1A1
SCHEMBL9633121 0.82 PLA2G4A (0.42) CYP1A2CYP2D6CYP2C19MTNR1AMTNR1B
SCHEMBL9633886 0.81 MAPT (0.49) CYP1A2CYP2D6CYP2C19MTNR1AMTNR1B
SCHEMBL9633804 0.81 NQO2 (0.48) MTNR1AMTNR1BNQO2MAPT
SCHEMBL9634189 0.81 PLA2G4A (0.41) CYP1A2CYP2D6CYP2C19MTNR1AMTNR1B
SCHEMBL10469188 0.80 CPT1A (0.49)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0337765-B1 ACYLSULFONAMIDE DERIVATIVES OF ALPHA-CARBOCYCLYLTOLUIC ACIDS USED AS LEUKOTRIENE ANTAGONISTS ICI AMERICAS INC. (US) 1992-10-14 EP disclosed
US-5095038-A Antiinflammatory, antiallergens ICI AMERICAS INC. (US) 1992-03-10 US disclosed
EP-0337765-A2 Acylsulfonamide derivatives of alpha-carbocyclyltoluic acids used as leukotriene antagonists ICI AMERICAS INC. (US) 1989-10-18 EP disclosed