SCHEMBL9634840

SCHEMBL9634840

CCOC(=O)CCCN1CCN(C(=O)OCc2ccccc2)CC1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 7/20 0.61
TMEM97 Q5BJF2 6/20 0.61
HRH2 P25021 3/20 0.61
HRH1 P35367 3/20 0.61
SLC6A2 P23975 2/20 0.61
CHRM1 P11229 1/20 0.61
HRH3 Q9Y5N1 1/20 0.61
HTR2A P28223 2/20 0.58
HTR1A P08908 1/20 0.58
CHRM5 P08912 1/20 0.58
ADRA1D P25100 1/20 0.58
HTR1B P28222 1/20 0.58
HTR2C P28335 1/20 0.58
HTR1E P28566 1/20 0.58
HTR2B P41595 1/20 0.58
SLC6A3 Q01959 1/20 0.58
L3MBTL1 Q9Y468 1/20 0.55
ADORA3 P0DMS8 1/20 0.54
HTR7 P34969 1/20 0.54
OPRM1 P35372 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29234166 0.89 HTT (0.56) SIGMAR1TMEM97HRH2HRH1SLC6A2
SCHEMBL21906828 0.87 L3MBTL1 (0.67) SIGMAR1TMEM97HRH2HRH1SLC6A2
SCHEMBL4904424 0.86 SIGMAR1 (0.57) SIGMAR1TMEM97HRH2HRH1SLC6A2
SCHEMBL9633964 0.86 MEN1 (0.57) SIGMAR1TMEM97HRH2HRH1HTR2A
SCHEMBL29207863 0.86 SIGMAR1 (0.52) SIGMAR1TMEM97HRH2HRH1SLC6A2
SCHEMBL29234309 0.86 HTT (0.55) SIGMAR1TMEM97HRH2HRH1SLC6A2
SCHEMBL5551353 0.85 KDM4E (0.62) SIGMAR1TMEM97HRH2HRH1SLC6A2
SCHEMBL27629467 0.85 SIGMAR1 (0.56) SIGMAR1TMEM97HRH2HRH1HTR2A
SCHEMBL19510869 0.85 KDM4E (0.62) SIGMAR1TMEM97HRH2HRH1SLC6A2
SCHEMBL7658562 0.84 L3MBTL1 (0.68) L3MBTL1NPC1RAB9ASMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0166509-B1 PHENOL DERIVATIVES IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1992-05-13 EP disclosed
US-4833135-A Antioestrogenic phenol derivatives IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1989-05-23 US disclosed
EP-0166509-A1 Phenol derivatives IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1986-01-02 EP disclosed