SCHEMBL9635627

SCHEMBL9635627

Cc1ccc2c(=O)cc(C#N)oc2c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.55
HPGD P15428 2/20 0.55
GAA P10253 1/20 0.55
POLB P06746 5/20 0.45
KMT2A Q03164 3/20 0.45
MAPT P10636 3/20 0.44
TP53 P04637 2/20 0.44
MAOB P27338 3/20 0.43
CSNK2A2 P19784 1/20 0.43
CSNK2B P67870 1/20 0.43
CSNK2A1 P68400 1/20 0.43
THRB P10828 1/20 0.40
HSD17B3 P37058 1/20 0.40
TNKS O95271 1/20 0.40
PARP1 P09874 1/20 0.40
TNKS2 Q9H2K2 1/20 0.40
PARP2 Q9UGN5 1/20 0.40
HTT P42858 1/20 0.40
CYP2A6 P11509 1/20 0.40
MEN1 O00255 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6961168 0.80 ALDH1A1 (0.55) ALDH1A1HPGDKMT2AMAPTTP53
SCHEMBL6956680 0.77 TNKS (0.58) ALDH1A1HPGDPOLBKMT2AMAPT
2,7-Dimethylchromone SCHEMBL7600130 0.77 ALDH1A1 (0.64) ALDH1A1HPGDGAAPOLBKMT2A
SCHEMBL9635524 0.76 CYP2A6 (0.37) POLBKMT2AMAOBTNKSCYP2A6
Selenium SCHEMBL30089787 0.76 TNKS (0.56) ALDH1A1HPGDPOLBKMT2AMAPT
SCHEMBL10257375 0.75 CYP2A6 (0.58) ALDH1A1GAAKMT2AMAPTMAOB
SCHEMBL29206959 0.72 HSD17B3 (0.73) ALDH1A1HPGDGAAKMT2AMAPT
SCHEMBL8025307 0.72 CYP2A6 (0.58) ALDH1A1MAOBCYP2A6
SCHEMBL7534248 0.71 MAPT (0.55) ALDH1A1HPGDPOLBMAPTTP53
SCHEMBL28050878 0.71 MAOB (0.77) ALDH1A1HPGDGAAKMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5082849-A Antiinflammatory agents or antiallergens AVENTIS PHARMACEUTICALS INC. 1992-01-21 US disclosed
EP-0434827-A4 QUINOLINYL-BENZOPYRAN DERIVATIVES AS ANTAGONISTS OF LEUKOTRIENE D 4? 1992-01-08 EP disclosed
EP-0434827-A1 QUINOLINYL-BENZOPYRAN DERIVATIVES AS ANTAGONISTS OF LEUKOTRIENE D 4? RORER INTERNATIONAL (HOLDINGS), INC. (US) 1991-07-03 EP disclosed
WO-1991001123-A2 QUINOLINYL-BENZOPYRAN DERIVATIVES AS ANTAGONISTS OF LEUKOTRIENE D¿4? RORER INTERNATIONAL (OVERSEAS) INC. (US) 1991-02-07 WO disclosed
US-4977162-A Quinolinyl-chromone derivatives and use for treatment of hypersensitive ailments RORER PHARMACEUTICAL CORPORATION (US) 1990-12-11 US disclosed