SCHEMBL9635668

SCHEMBL9635668

C=CCOc1ccc(-c2nc3cnccc3[nH]2)c(O)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
NPSR1 Q6W5P4 1/20 0.40
MAPT P10636 2/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
HPGD P15428 2/20 0.38
GAA P10253 2/20 0.38
MAOA P21397 2/20 0.38
ALDH1A1 P00352 1/20 0.38
AMY1A P0DUB6 1/20 0.38
MGAM O43451 1/20 0.37
SI P14410 1/20 0.37
MGAM2 Q2M2H8 1/20 0.37
SLC5A1 P13866 1/20 0.34
SLC5A2 P31639 1/20 0.34
KDM4E B2RXH2 1/20 0.34
KDM4A O75164 1/20 0.34
KDM5C P41229 1/20 0.34
KDM4D Q6B0I6 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9635742 0.89 PDE5A (0.39) LMNASMN1; SMN2NPSR1MAPTMEN1
SCHEMBL9635925 0.86 PDE5A (0.47) LMNASMN1; SMN2NPSR1MAPTMEN1
SCHEMBL9634609 0.85 CDK4 (0.40) SMN1; SMN2NPSR1MAPTMEN1KMT2A
SCHEMBL9634469 0.85 PDE5A (0.41) LMNASMN1; SMN2NPSR1MAPTMEN1
SCHEMBL9635794 0.85 PDE5A (0.40) LMNASMN1; SMN2NPSR1MAPTMEN1
SCHEMBL9636522 0.85 MAOA (0.38) LMNASMN1; SMN2NPSR1MAPTMEN1
SCHEMBL9634973 0.85 CBFB (0.46) LMNASMN1; SMN2NPSR1MAPTMEN1
SCHEMBL9635832 0.84 CHEK2 (0.42) NPSR1MAPTMEN1KMT2AHPGD
SCHEMBL9634904 0.83 PDE5A (0.39) LMNASMN1; SMN2NPSR1MAPTMEN1
SCHEMBL9636206 0.83 PDE5A (0.37) LMNASMN1; SMN2NPSR1MAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5104881-A 2-ARYLIMIDAZOPYRIDINES MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1992-04-14 US disclosed
US-4616090-A 2-arylimidazopyridines intermediates MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1986-10-07 US disclosed
EP-0072926-B1 2-ARYLIMIDAZOPYRIDINES MERCK PATENT GmbH (DE) 1986-09-24 EP disclosed
EP-0072926-A1 2-Arylimidazopyridines MERCK PATENT GmbH (DE) 1983-03-02 EP disclosed