SCHEMBL9637314

SCHEMBL9637314

C=C1S[C@H]2[C@@H](Br)C(=O)N2C(C(=O)OC(c2ccccc2)c2ccccc2)=C1C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.38
ESR2 Q92731 1/20 0.38
ELANE P08246 8/20 0.36
ALDH1A1 P00352 6/20 0.35
HPGD P15428 4/20 0.35
HSD17B10 Q99714 3/20 0.35
KMT2A Q03164 3/20 0.35
MAPT P10636 3/20 0.35
CYP3A4 P08684 2/20 0.35
SLC15A2 Q16348 2/20 0.35
TDP1 Q9NUW8 2/20 0.35
BLM P54132 1/20 0.35
CYP2C19 P33261 1/20 0.35
MAPK1 P28482 1/20 0.35
ADRA1A P35348 1/20 0.35
HTR2B P41595 1/20 0.35
POLB P06746 1/20 0.34
KDM4E B2RXH2 3/20 0.32
LMNA P02545 1/20 0.32
PTGS1 P23219 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9635961 0.87 ELANE (0.36) ESR1ESR2ELANEALDH1A1HPGD
SCHEMBL9635856 0.79 ELANE (0.45) ESR1ESR2ELANEALDH1A1HPGD
SCHEMBL8669679 0.79 ALDH1A1 (0.51) ESR1ALDH1A1HPGDHSD17B10KMT2A
SCHEMBL8669680 0.79 ALDH1A1 (0.51) ESR1ALDH1A1HPGDHSD17B10KMT2A
SCHEMBL8667178 0.77 ESR1 (0.34) ESR1ESR2ELANEALDH1A1HPGD
SCHEMBL8667176 0.77 ESR1 (0.34) ESR1ESR2ELANEALDH1A1HPGD
SCHEMBL9755490 0.77 MEN1 (0.31) ESR1HSD17B10KMT2AMAPTSLC15A2
SCHEMBL9755501 0.76 ELANE (0.39) ELANECTDSP1
SCHEMBL9755503 0.76 ELANE (0.39) ELANECTDSP1
SCHEMBL11360226 0.72 PTGS1 (0.57) ESR1ELANEHPGDHSD17B10KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0494914-A1 NOVEL 2-SPIROCYCLOPROPYL CEPHALOSPORIN SULFONE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF SYNPHAR LABORATORIES INC. (CA) 1992-07-22 EP disclosed