SCHEMBL9639712

SCHEMBL9639712

CCNc1cccnc1N1CCN(C(C)C(=O)OCc2ccccc2)CC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.46
LMNA P02545 4/20 0.42
SMN1; SMN2 Q16637 4/20 0.42
MAPT P10636 3/20 0.42
USP2 O75604 2/20 0.42
MEN1 O00255 1/20 0.42
PABPC1 P11940 1/20 0.42
TSHR P16473 1/20 0.42
CASP1 P29466 1/20 0.42
KMT2A Q03164 1/20 0.42
EIF4H Q15056 1/20 0.42
TP53 P04637 1/20 0.42
GFER P55789 1/20 0.42
TGM2 P21980 1/20 0.41
CSNK1A1 P48729 2/20 0.41
CHIA Q9BZP6 1/20 0.40
ALDH1A1 P00352 2/20 0.40
CAPN1 P07384 1/20 0.39
CTSS P25774 1/20 0.39
GRIN2B Q13224 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9640895 0.85 PARP1 (0.52) PARP1KMT2ACHIAMAPK1
Hydrochloric Acid SCHEMBL9755172 0.84 PARP1 (0.51) PARP1KMT2ACHIAMAPK1
E1501 SCHEMBL9639366 0.80 PARP1 (0.46) PARP1CSNK1A1ALDH1A1GRIN2BL3MBTL1
SCHEMBL9640454 0.79 PARP1 (0.45) PARP1TSHRCSNK1A1GRIN2BL3MBTL1
SCHEMBL9755185 0.78 PARP1 (0.51) PARP1MEN1KMT2ATP53CHIA
SCHEMBL9639396 0.77 PARP1 (0.48) PARP1MEN1KMT2ATP53CHIA
Acetic Acid SCHEMBL9639371 0.77 HTR3E (0.53) PARP1LMNASMN1; SMN2MAPTMEN1
Propionic Acid SCHEMBL9640459 0.76 HTR3E (0.52) PARP1LMNASMN1; SMN2MAPTCHIA
SCHEMBL8917544 0.74 HDAC1 (0.49) SMN1; SMN2MEN1KMT2ATGM2GRIN2B
SCHEMBL9639717 0.73 PARP1 (0.45) PARP1MEN1TSHRKMT2ACHIA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0496746-A1 PHARMACEUTICALLY ACTIVE AMINO-SUBSTITUTED HETEROARYL AMINES THE UPJOHN COMPANY (US) 1992-08-05 EP claimed
WO-1991006542-A1 PHARMACEUTICALLY ACTIVE AMINO-SUBSTITUTED HETEROARYL AMINES THE UPJOHN COMPANY (US) 1991-05-16 WO claimed
WO-1991006542-A1 PHARMACEUTICALLY ACTIVE AMINO-SUBSTITUTED HETEROARYL AMINES THE UPJOHN COMPANY (US) 1991-05-16 WO disclosed