SCHEMBL9639717

SCHEMBL9639717

CCNc1cccnc1N1CCN(OC(=O)CCCc2ccccc2)CC1

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.45
KMT2A Q03164 3/20 0.42
MEN1 O00255 2/20 0.42
TSHR P16473 1/20 0.41
HSD17B10 Q99714 1/20 0.41
CHIA Q9BZP6 1/20 0.39
ALDH1A1 P00352 2/20 0.38
GAA P10253 1/20 0.38
HRH4 Q9H3N8 1/20 0.37
AR P10275 1/20 0.37
MAPK1 P28482 1/20 0.37
FAAH O00519 1/20 0.36
PLAAT3 P53816 1/20 0.36
PLAAT5 Q96KN8 1/20 0.36
PLAAT2 Q9NWW9 1/20 0.36
PLAAT4 Q9UL19 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9639375 0.94 PARP1 (0.46) PARP1KMT2AMEN1TSHRHSD17B10
SCHEMBL9639398 0.88 PARP1 (0.48) PARP1KMT2AMEN1TSHRCHIA
SCHEMBL9755187 0.87 PARP1 (0.50) PARP1KMT2AMEN1TSHRCHIA
SCHEMBL9640899 0.84 PARP1 (0.52) PARP1KMT2AMEN1CHIAGAA
Hydrochloric Acid SCHEMBL9755174 0.83 PARP1 (0.51) PARP1KMT2AMEN1CHIAGAA
Acetic Acid SCHEMBL9639371 0.76 HTR3E (0.53) PARP1KMT2AMEN1ALDH1A1MAPK1
Propionic Acid SCHEMBL9640459 0.75 HTR3E (0.52) PARP1CHIAALDH1A1MAPK1
SCHEMBL9639544 0.74 PARP1 (0.50) PARP1CHIAALDH1A1
SCHEMBL9755222 0.73 PARP1 (0.52) PARP1KMT2AMEN1CHIAALDH1A1
SCHEMBL9639712 0.73 PARP1 (0.46) PARP1KMT2AMEN1TSHRCHIA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0496746-A1 PHARMACEUTICALLY ACTIVE AMINO-SUBSTITUTED HETEROARYL AMINES THE UPJOHN COMPANY (US) 1992-08-05 EP claimed
WO-1991006542-A1 PHARMACEUTICALLY ACTIVE AMINO-SUBSTITUTED HETEROARYL AMINES THE UPJOHN COMPANY (US) 1991-05-16 WO claimed
EP-0496746-A1 PHARMACEUTICALLY ACTIVE AMINO-SUBSTITUTED HETEROARYL AMINES THE UPJOHN COMPANY (US) 1992-08-05 EP disclosed
WO-1991006542-A1 PHARMACEUTICALLY ACTIVE AMINO-SUBSTITUTED HETEROARYL AMINES THE UPJOHN COMPANY (US) 1991-05-16 WO disclosed