SCHEMBL9640991

SCHEMBL9640991

CC(Cc1ccccc1)NC(C)C(O)c1ccccc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 4/20 0.64
ADRA1A P35348 5/20 0.60
CYP2D6 P10635 5/20 0.60
CYP2C19 P33261 5/20 0.60
CYP1A2 P05177 4/20 0.60
ADRA2C P18825 3/20 0.60
HTR2A P28223 3/20 0.60
TSHR P16473 3/20 0.60
HTR1A P08908 3/20 0.60
SLC6A2 P23975 3/20 0.60
OPRM1 P35372 3/20 0.60
DRD3 P35462 3/20 0.60
SLC6A3 Q01959 3/20 0.60
KCNH2 Q12809 3/20 0.60
CYP3A4 P08684 2/20 0.60
NFKB1 P19838 2/20 0.60
ADRB2 P07550 2/20 0.60
ADRB1 P08588 2/20 0.60
ADRA2B P18089 2/20 0.60
OPRK1 P41145 2/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ephedrine SCHEMBL16196643 0.83 ADRA1A (0.71) SIGMAR1ADRA1ACYP2D6CYP2C19CYP1A2
Pseudoephedrine SCHEMBL16601218 0.83 ADRA1A (0.71) SIGMAR1ADRA1ACYP2D6CYP2C19CYP1A2
SCHEMBL28002406 0.80 SIGMAR1 (0.63) SIGMAR1CYP2D6CYP1A2TSHRCYP3A4
SCHEMBL21243273 0.79 SIGMAR1 (0.73) SIGMAR1CYP2D6CYP1A2TSHRSLC6A2
SCHEMBL5270097 0.79 LMNA (0.79) SIGMAR1ADRA1ACYP2D6CYP2C19CYP1A2
SCHEMBL7637484 0.79 LMNA (0.79) SIGMAR1ADRA1ACYP2D6CYP2C19CYP1A2
SCHEMBL7785516 0.79 LMNA (0.79) SIGMAR1ADRA1ACYP2D6CYP2C19CYP1A2
SCHEMBL9322567 0.78 SIGMAR1 (1.00) SIGMAR1ADRA1ACYP2D6CYP1A2ADRA2C
SCHEMBL28073509 0.78 SIGMAR1 (0.72) SIGMAR1ADRA1ACYP2D6CYP1A2ADRA2C
SCHEMBL12573499 0.77 ADRA1A (0.67) ADRA1ACYP2D6CYP2C19CYP1A2ADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0290122-B1 MORPHOLINE DERIVATIVES AND THEIR USE BEECHAM GROUP PLC (GB) 1992-12-23 EP disclosed
US-5082840-A Animal growth regulators BEECHAM GROUP P.L.C. (GB) 1992-01-21 US disclosed
US-4914202-A FOR IMPROVING FEED EFFICIENCY IN LIVESTOCK BEECHAM GROUP P.L.C. (GB) 1990-04-03 US disclosed
EP-0290122-A1 Morpholine derivatives and their use BEECHAM GROUP PLC (GB) 1988-11-09 EP disclosed