SCHEMBL9644656

SCHEMBL9644656

COc1cc(N)c(Cl)cc1C(=O)NC1CC2CCCCN2C1

nearest known ligand 0.70

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
HTR4 Q13639 7/20 0.68
DRD2 P14416 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10553783 0.92 HTR4 (0.65) HTR4DRD2
SCHEMBL9645517 0.92 HTR4 (0.73) HTR4DRD2
SCHEMBL11456465 0.92 HTR4 (0.70) HTR4DRD2
SCHEMBL11397386 0.89 DRD4 (0.72) HTR4
SCHEMBL11002126 0.89 HTR4 (0.74) HTR4DRD2
SCHEMBL11457053 0.86 HTR4 (0.69) HTR4DRD2
SCHEMBL9644709 0.85 DRD4 (0.67) HTR4
Fumaric Acid SCHEMBL11580335 0.84 DRD4 (0.65) HTR4DRD2
Fumaric Acid SCHEMBL11580339 0.84 DRD4 (0.65) HTR4DRD2
SCHEMBL8722682 0.81 HTR4 (1.00) HTR4DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0327335-B1 ARYLAMIDO(AND ARYLTHIOAMIDO)-AZABICYCLOALKANES FOR ENHANCING MEMORY OR CORRECTING MEMORY DEFICIENCY SYNTHELABO (FR) 1992-10-14 EP disclosed
US-4863919-A Method of enhancing memory or correcting memory deficiency with arylamido(and arylthiomido)-azabicycloalkanes A. H. ROBINS COMPANY, INCORPORATED (US) 1989-09-05 US disclosed
EP-0327335-A1 Arylamido(and arylthioamido)-azabicycloalkanes for enhancing memory or correcting memory deficiency SYNTHELABO (FR) 1989-08-09 EP disclosed
EP-0190920-A2 Method of enhancing memory or correcting memory deficiency with arylamido (and arylthioamido)azabicycloalkanes SYNTHELABO (FR) 1986-08-13 EP disclosed
US-4605652-A ALZHEIMER'S DISEASE; SENILITY A. H. ROBINS COMPANY, INC. (US) 1986-08-12 US disclosed
US-4213983-A Treating gastro-intestinal disorders and emesis with n-(heterocyclic substituted) benzamides BEECHAM GROUP LIMITED (GB) 1980-07-22 US disclosed