SCHEMBL9645173

SCHEMBL9645173

CC(C)(C)OC(=O)Nc1ccc2c(=O)n(Cc3cccnc3)[nH]c2c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 2/20 0.54
NAMPT P43490 2/20 0.46
ALDH1A1 P00352 3/20 0.41
KMT2A Q03164 2/20 0.41
MEN1 O00255 1/20 0.41
LMNA P02545 1/20 0.41
MAPT P10636 1/20 0.41
HTT P42858 1/20 0.41
CYP17A1 P05093 1/20 0.41
CYP3A4 P08684 1/20 0.40
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA9 Q16790 1/20 0.39
KDM4E B2RXH2 2/20 0.39
GLA P06280 1/20 0.39
GAA P10253 1/20 0.39
HPGD P15428 1/20 0.39
TSHR P16473 1/20 0.39
HSD17B10 Q99714 1/20 0.39
PKM P14618 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9647127 0.80 ALOX5 (0.53) ALOX5NAMPTALDH1A1LMNAKDM4E
SCHEMBL9669683 0.80 ALOX5 (0.54) ALOX5NAMPTALDH1A1CYP3A4KDM4E
SCHEMBL9646389 0.74 ALOX5 (0.70) ALOX5KMT2AMEN1CYP3A4PKM
SCHEMBL916112 0.74 NAMPT (0.48) NAMPTALDH1A1KMT2AMEN1LMNA
SCHEMBL9596545 0.72 ALOX5 (1.00) ALOX5KDM4EPKM
SCHEMBL17790711 0.70 PARP1 (0.53) NAMPTKMT2AMEN1CYP17A1CYP3A4
SCHEMBL29457342 0.69 NAMPT (0.80) NAMPTLMNAHTTCYP3A4KDM4E
SCHEMBL349933 0.69 NAMPT (0.80) NAMPTLMNAHTTCYP3A4KDM4E
SCHEMBL25468287 0.68 NAMPT (0.40) NAMPTMAPTCYP17A1CYP3A4GAA
SCHEMBL5716528 0.67 CYP3A4 (0.44) NAMPTALDH1A1CYP3A4PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5173496-A Antiinflammatory agents ICI PHARMA (FR) 1992-12-22 US disclosed