SCHEMBL9645835

SCHEMBL9645835

O=C1CC=CN(c2ccc3ccccc3n2)N1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.44
KDM4E B2RXH2 6/20 0.44
HTR3E A5X5Y0 2/20 0.44
HTR3B O95264 2/20 0.44
CYP1A2 P05177 2/20 0.44
HTR3A P46098 2/20 0.44
HTR3D Q70Z44 2/20 0.44
HTR3C Q8WXA8 2/20 0.44
CYP3A4 P08684 2/20 0.44
HSD17B10 Q99714 2/20 0.44
USP2 O75604 2/20 0.44
TDP1 Q9NUW8 2/20 0.44
HTR1A P08908 2/20 0.44
ADRB1 P08588 1/20 0.44
HTR2C P28335 1/20 0.44
MAPK1 P28482 1/20 0.44
SLC6A4 P31645 1/20 0.44
HTR7 P34969 1/20 0.44
HTT P42858 1/20 0.44
HTR6 P50406 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7604149 0.75 CRBN (0.50) ALDH1A1KDM4ECYP1A2HSD17B10MAPK1
SCHEMBL3781498 0.68 KDM4E (0.55) ALDH1A1KDM4EHTR3EHTR3BCYP1A2
SCHEMBL9645827 0.68 ALOX5 (0.54) ALDH1A1KDM4EHTR3EHTR3BCYP1A2
SCHEMBL3798927 0.66 RECQL (0.51) ALDH1A1KDM4EHTR3EHTR3BCYP1A2
SCHEMBL10792966 0.64 KMT2A (0.48) ALDH1A1KDM4EHTR3EHTR3BCYP1A2
SCHEMBL5742495 0.64 USP2 (0.48) ALDH1A1KDM4EHTR3EHTR3BCYP1A2
SCHEMBL10609190 0.64 HRH3 (0.63) ALDH1A1KDM4EHTR3EHTR3BCYP1A2
SCHEMBL11548784 0.63 HTR1A (0.51) ALDH1A1KDM4EHTR3EHTR3BCYP1A2
SCHEMBL30046397 0.63 HTR1A (0.51) ALDH1A1KDM4EHTR3EHTR3BCYP1A2
SCHEMBL7471396 0.63 ALDH1A1 (0.61) ALDH1A1KDM4EHTR3EHTR3BCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5086052-A Antiarthritic, antiallergens, antiinflammatory agents; also for asthma and psoriasis ABBOTT LABORATORIES (US) 1992-02-04 US disclosed
EP-0299449-A2 Pyridazinone, triazinone and oxapyridazinone lipoxygenase inhibiting compounds ABBOTT LABORATORIES (US) 1989-01-18 EP disclosed