SCHEMBL9650010

SCHEMBL9650010

COc1ccc(-c2cn3c(=O)n(Cc4ccccc4)c4ccccc4c3n2)cc1OC

nearest known ligand 0.68

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 0.52
ADORA2A P29274 1/20 0.52
ADORA1 P30542 1/20 0.52
PDE4A P27815 3/20 0.50
PDE4B Q07343 3/20 0.50
PDE4C Q08493 3/20 0.50
PDE4D Q08499 3/20 0.50
KMT2A Q03164 1/20 0.48
ALDH1A1 P00352 2/20 0.47
MAPT P10636 2/20 0.47
PTGDR2 Q9Y5Y4 1/20 0.47
PDE3B Q13370 1/20 0.44
PDE3A Q14432 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.43
PARP1 P09874 1/20 0.43
TP53 P04637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9649859 0.81 TSPO (0.55) ADORA3ADORA2AADORA1TP53
SCHEMBL4648097 0.73 PDE4A (0.49) PDE4APDE4BPDE4CPDE4DKMT2A
SCHEMBL4013052 0.71 MAP3K11 (0.71) PDE4APDE4BPDE4CPDE4D
SCHEMBL9213247 0.70 ALDH1A1 (0.48) KMT2AALDH1A1MAPT
SCHEMBL11576284 0.70 PDE4A (0.55) PDE4APDE4BPDE4CPDE4DALDH1A1
SCHEMBL28127173 0.69 PDE4A (0.50) PDE4APDE4BPDE4CPDE4DKMT2A
Hydrochloric Acid SCHEMBL11578577 0.69 PDE4A (0.54) PDE4APDE4BPDE4CPDE4DALDH1A1
SCHEMBL28127167 0.69 MCL1 (0.58) PDE4APDE4BPDE4CPDE4DALDH1A1
SCHEMBL9649918 0.68 CYP1A2 (0.56) KMT2AALDH1A1
SCHEMBL9217903 0.68 TSPO (0.59) ALDH1A1MAPTSMN1; SMN2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5128338-A Cardiovascular disorders ADIR ET COMPAGNIE (FR) 1992-07-07 US disclosed