SCHEMBL9652003

SCHEMBL9652003

CC(C)(C)N(NC(=O)c1c(F)cccc1F)C(=O)c1cccs1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
POLB P06746 1/20 0.43
TSHR P16473 1/20 0.42
HPGD P15428 1/20 0.41
NPC1 O15118 2/20 0.40
ABCB1 P08183 1/20 0.40
HDAC1 Q13547 1/20 0.40
CASP3 P42574 1/20 0.39
SENP8 Q96LD8 1/20 0.39
SENP7 Q9BQF6 1/20 0.39
SENP6 Q9GZR1 1/20 0.39
ALDH1A1 P00352 1/20 0.39
CES2 O00748 1/20 0.39
CES1 P23141 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9651998 0.90 RAB9A (0.46) RAB9ACYP3A4CYP2C9POLBTSHR
SCHEMBL9496544 0.83 POLB (0.51) CYP3A4CYP2C9POLBHPGDABCB1
SCHEMBL8180270 0.80 POLB (0.68) RAB9ACYP3A4CYP2C9POLBNPC1
SCHEMBL9714560 0.79 POLB (0.70) CYP3A4CYP2C9POLBABCB1
SCHEMBL9651954 0.78 NPC1 (0.58) RAB9ACYP3A4CYP2C9POLBHPGD
SCHEMBL9651981 0.78 ABCB1 (0.69) CYP3A4CYP2C9POLBABCB1ALDH1A1
SCHEMBL10718940 0.77 CYP3A4 (0.56) CYP3A4CYP2C9POLBABCB1
SCHEMBL9651937 0.77 RAB9A (0.57) RAB9ACYP3A4CYP2C9POLBNPC1
SCHEMBL8172543 0.75 POLB (0.68) RAB9ACYP3A4CYP2C9POLBTSHR
SCHEMBL10747617 0.74 ABCB1 (0.46) ABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0261755-B1 FIVE-MEMBERED HETEROCYCLIC DERIVATIVES OF N'-SUBSTITUTED-N,N'-DIACYLHYDRAZINES ROHM AND HAAS COMPANY (US) 1992-12-16 EP disclosed