SCHEMBL9651998

SCHEMBL9651998

CC(C)(C)N(NC(=O)c1cccs1)C(=O)c1c(F)cccc1F

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 5/20 0.46
TSHR P16473 1/20 0.45
HPGD P15428 1/20 0.44
NPC1 O15118 4/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
HDAC1 Q13547 1/20 0.43
POLB P06746 1/20 0.43
ALDH1A1 P00352 2/20 0.42
CASP3 P42574 1/20 0.42
SENP8 Q96LD8 1/20 0.42
SENP7 Q9BQF6 1/20 0.42
SENP6 Q9GZR1 1/20 0.42
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
TP53 P04637 1/20 0.40
MAPT P10636 1/20 0.40
PKM P14618 1/20 0.40
NFKB1 P19838 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9652003 0.90 RAB9A (0.43) RAB9ATSHRHPGDNPC1CYP3A4
SCHEMBL9496544 0.83 POLB (0.51) HPGDCYP3A4CYP2C9POLBSMN1; SMN2
SCHEMBL8172543 0.80 POLB (0.68) RAB9ATSHRNPC1CYP3A4CYP2C9
SCHEMBL9714565 0.79 POLB (0.70) CYP3A4CYP2C9POLB
SCHEMBL9651949 0.78 NPC1 (0.58) RAB9ATSHRHPGDNPC1CYP3A4
SCHEMBL9651986 0.78 ABCB1 (0.65) CYP3A4CYP2C9POLBALDH1A1MEN1
SCHEMBL9651939 0.77 RAB9A (0.57) RAB9ATSHRHPGDNPC1CYP3A4
SCHEMBL8180270 0.75 POLB (0.68) RAB9ANPC1CYP3A4CYP2C9POLB
SCHEMBL9651153 0.74 MAPT (0.60) HPGDCYP3A4CYP2C9POLBMEN1
SCHEMBL9714560 0.73 POLB (0.70) CYP3A4CYP2C9POLBSMN1; SMN2ABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0261755-B1 FIVE-MEMBERED HETEROCYCLIC DERIVATIVES OF N'-SUBSTITUTED-N,N'-DIACYLHYDRAZINES ROHM AND HAAS COMPANY (US) 1992-12-16 EP disclosed