SCHEMBL9656015

SCHEMBL9656015

N=C(N)Nc1nnc(-c2ccccc2C(F)(F)F)s1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 10/20 0.43
RAB9A P51151 9/20 0.43
RXFP1 Q9HBX9 2/20 0.43
ALDH1A1 P00352 6/20 0.42
KDM4E B2RXH2 6/20 0.42
SMN1; SMN2 Q16637 5/20 0.42
HSD11B1 P28845 1/20 0.41
HPGD P15428 4/20 0.40
LMNA P02545 1/20 0.40
WNT3A P56704 1/20 0.40
HSD17B10 Q99714 4/20 0.39
TP53 P04637 2/20 0.39
CYP1A2 P05177 1/20 0.39
AHR P35869 1/20 0.39
PKM P14618 1/20 0.39
CASP3 P42574 1/20 0.39
SENP8 Q96LD8 1/20 0.39
SENP7 Q9BQF6 1/20 0.39
SENP6 Q9GZR1 1/20 0.39
VCP P55072 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9656027 0.99 NPC1 (0.42) NPC1RAB9ARXFP1ALDH1A1KDM4E
SCHEMBL9656920 0.84 HSD11B1 (0.46) NPC1RAB9ARXFP1ALDH1A1KDM4E
SCHEMBL9656308 0.82 HSD11B1 (0.47) NPC1RAB9ARXFP1ALDH1A1KDM4E
Hydrochloric Acid SCHEMBL11564981 0.81 ALDH1A1 (0.47) NPC1RAB9ARXFP1ALDH1A1KDM4E
Hydrochloric Acid SCHEMBL9656358 0.76 KDM4E (0.41) NPC1RAB9ARXFP1ALDH1A1KDM4E
Hydrochloric Acid SCHEMBL9264701 0.75 MAPT (0.48) RAB9ARXFP1ALDH1A1SMN1; SMN2MEN1
SCHEMBL9656933 0.75 HSD11B1 (0.41) NPC1RAB9AALDH1A1KDM4ESMN1; SMN2
SCHEMBL9654561 0.74 PTGS1 (0.45) NPC1RAB9ARXFP1ALDH1A1KDM4E
SCHEMBL6678346 0.74 ALDH1A1 (0.64) RAB9AALDH1A1KDM4ESMN1; SMN2HSD11B1
SCHEMBL2442712 0.72 HSD11B1 (0.54) ALDH1A1HSD11B1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0288185-B1 THIADIAZOLE GUANIDINES RECKITT AND COLMAN PRODUCTS LIMITED (GB) 1992-08-19 EP claimed
US-4786627-A ANTI-CONVULSANTS RECKITT & COLMAN PRODUCTS LIMITED (GB) 1988-11-22 US claimed
EP-0288185-A1 Thiadiazole guanidines RECKITT AND COLMAN PRODUCTS LIMITED (GB) 1988-10-26 EP claimed