SCHEMBL9656646

SCHEMBL9656646

Cc1[nH]cnc1CC(=O)C(OC(=O)/C=C\C(=O)OC(C(=O)Cc1nc[nH]c1C)c1cc2ccccc2n1C)c1cc2ccccc2n1C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRR1 P24046 1/20 0.41
HTR3A P46098 3/20 0.38
HTR3E A5X5Y0 2/20 0.38
HTR3B O95264 2/20 0.38
HTR3D Q70Z44 2/20 0.38
HTR3C Q8WXA8 2/20 0.38
MCL1 Q07820 1/20 0.35
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
ADRA2C P18825 1/20 0.34
HTR2A P28223 1/20 0.34
HTR2C P28335 1/20 0.34
ADRA1A P35348 1/20 0.34
HTR2B P41595 1/20 0.34
KCNH2 Q12809 1/20 0.34
CTSL P07711 1/20 0.34
CTSS P25774 1/20 0.34
CTSK P43235 1/20 0.34
CASP6 P55212 1/20 0.34
UTS2R Q9UKP6 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fumaric Acid SCHEMBL9656647 0.75 GABRR1 (0.43) GABRR1HTR3AHTR3EHTR3BHTR3D
Maleic Acid SCHEMBL9656644 0.75 GABRR1 (0.43) GABRR1HTR3AHTR3EHTR3BHTR3D
SCHEMBL7274925 0.73 HTR3E (0.43) GABRR1HTR3AHTR3EHTR3BHTR3D
SCHEMBL7272916 0.73 HTR3E (0.46) GABRR1HTR3AHTR3EHTR3BHTR3D
SCHEMBL7297785 0.72 HTR3E (0.42) GABRR1HTR3AHTR3EHTR3BHTR3D
SCHEMBL7265491 0.71 HTR3E (0.41) GABRR1HTR3AHTR3EHTR3BHTR3D
Fumaric Acid SCHEMBL7323811 0.71 HTR3E (0.44) GABRR1HTR3AHTR3EHTR3BHTR3D
Maleic Acid SCHEMBL9656645 0.70 HTR3E (0.53) GABRR1HTR3AHTR3EHTR3BHTR3D
Fumaric Acid SCHEMBL9668452 0.70 HTR3E (0.53) GABRR1HTR3AHTR3EHTR3BHTR3D
SCHEMBL9656120 0.65 MCL1 (0.35) HTR3AMCL1CYP1A2CYP3A4ADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5084474-A Antagonist of 5-hydroxytryptamine receptors on nerves and useful for treatment of psychotic disorders, anxiety, and nausea and vomiting, compounds of imidazole GLAXO GROUP LIMITED (GB) 1992-01-28 US disclosed