SCHEMBL9656805

SCHEMBL9656805

Cc1nc(CC(O)(P(=O)(O)O)P(=O)(O)O)cs1

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
FDPS P14324 10/20 0.45
SMN1; SMN2 Q16637 5/20 0.41
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
TDP1 Q9NUW8 1/20 0.41
ALDH1A1 P00352 2/20 0.40
MAPT P10636 1/20 0.40
HPGD P15428 1/20 0.39
POLB P06746 1/20 0.38
LMNA P02545 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
KMT2A Q03164 1/20 0.38
BTN3A1 O00481 1/20 0.37
PDE3A Q14432 1/20 0.37
GAA P10253 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10624905 0.84 SMN1; SMN2 (0.45) FDPSSMN1; SMN2NPC1RAB9ATDP1
SCHEMBL3556536 0.75 PGK1 (0.47) SMN1; SMN2NPC1RAB9ATDP1ALDH1A1
SCHEMBL9658614 0.75 FDPS (0.44) FDPSSMN1; SMN2NPC1RAB9ATDP1
SCHEMBL1912692 0.72 GAA (0.44) SMN1; SMN2NPC1RAB9ATDP1ALDH1A1
SCHEMBL4120827 0.72 PKM (0.42) SMN1; SMN2NPC1RAB9ATDP1ALDH1A1
SCHEMBL13544288 0.71 GAA (0.43) SMN1; SMN2NPC1RAB9ATDP1ALDH1A1
SCHEMBL1107640 0.69 PKM (0.48) SMN1; SMN2NPC1RAB9ATDP1ALDH1A1
SCHEMBL9657444 0.69 FDPS (0.47) FDPSBTN3A1PDE3A
SCHEMBL4134899 0.69 PKM (0.45) SMN1; SMN2NPC1RAB9ATDP1ALDH1A1
SCHEMBL10974541 0.69 SMN1; SMN2 (0.53) SMN1; SMN2NPC1RAB9ATDP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0258618-B1 DIPHOSPHONIC ACID DERIVATIVES, PROCESS FOR THEIR PREPARATION AND MEDICINES CONTAINING THOSE COMPOUNDS Roche Diagnostics GmbH (DE) 1992-05-06 EP disclosed
US-4777163-A BONE DISORDERS, RHEUMATIC DISEASES BOEHRINGER MANNHEIM GMBH (DE) 1988-10-11 US disclosed
EP-0258618-A2 Diphosphonic acid derivatives, process for their preparation and medicines containing those compounds Roche Diagnostics GmbH (DE) 1988-03-09 EP disclosed