SCHEMBL9662002

SCHEMBL9662002

CCn1cc(Br)nc(N)c1=O

nearest known ligand 0.34

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 1/20 0.34
CCNB1 P14635 1/20 0.34
CCNE1 P24864 1/20 0.34
CDK2 P24941 1/20 0.34
ADORA1 P30542 3/20 0.33
ADORA2A P29274 3/20 0.33
BRD4 O60885 2/20 0.33
ADORA3 P0DMS8 1/20 0.33
ADORA2B P29275 1/20 0.33
PI4KA P42356 1/20 0.32
PI4K2B Q8TCG2 1/20 0.32
PI4K2A Q9BTU6 1/20 0.32
PI4KB Q9UBF8 1/20 0.32
ALDH1A1 P00352 1/20 0.32
EEF2K O00418 1/20 0.31
ALPL P05186 2/20 0.31
PLAA Q9Y263 1/20 0.31
TSHR P16473 1/20 0.30
ALPG P10696 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL925383 0.81 BRD4 (0.35) BRD4ALDH1A1ALPLPLAAALPG
SCHEMBL13694927 0.79 ALPL (0.34) BRD4ALDH1A1ALPLPLAAALPG
SCHEMBL13512616 0.75 AURKA (0.40) ADORA1ADORA2ABRD4ADORA2B
SCHEMBL12401883 0.71 TLR8 (0.52) ADORA1ADORA2ABRD4ADORA3ALDH1A1
SCHEMBL15573640 0.71
SCHEMBL23213724 0.65 ALPL (0.32) ALDH1A1ALPLPLAAALPG
SCHEMBL19924655 0.65 BRD4 (0.69) BRD4
SCHEMBL11718699 0.64 EP300 (0.43) CDK1CCNB1CCNE1CDK2ADORA1
SCHEMBL5201162 0.64 CDK1 (0.35) CDK1CCNB1CCNE1CDK2ADORA1
SCHEMBL8178792 0.64 CNR2 (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0262096-B1 AMINOPYRAZINONES AND AMINOTRIAZINONES CIBA-GEIGY AG (CH) 1992-01-02 EP disclosed
US-4920223-A Herbicides, plant growth regulators CIBA-GEIGY CORPORATION (US) 1990-04-24 US disclosed
US-4871853-A HERBICIDE INTERMEDIATES CIBA-GEIGY CORPORATION (US) 1989-10-03 US disclosed
US-4795486-A HERBICIDES, PLANT GROWTH REGULATORS CIBA-GEIGY CORPORATION, 444 SAW MILL RIVER ROAD, ARDSLEY, NEW YORK 10502 A NY CORP. 1989-01-03 US disclosed
EP-0262096-A1 Aminopyrazinones and aminotriazinones CIBA-GEIGY AG (CH) 1988-03-30 EP disclosed