SCHEMBL9664008

SCHEMBL9664008

CC(=O)CC(=O)c1ccc2ccccc2n1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.60
MAPT P10636 2/20 0.60
GAA P10253 1/20 0.60
MGAM O43451 1/20 0.58
HDAC8 Q9BY41 1/20 0.57
KDM4C Q9H3R0 1/20 0.54
HPGD P15428 2/20 0.54
CNR2 P34972 3/20 0.53
SMN1; SMN2 Q16637 5/20 0.53
RAB9A P51151 5/20 0.53
NFKB1 P19838 3/20 0.53
NFKB2 Q00653 3/20 0.53
RELA Q04206 3/20 0.53
NPC1 O15118 4/20 0.50
KDM4E B2RXH2 3/20 0.50
TP53 P04637 2/20 0.50
POLB P06746 1/20 0.50
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
RECQL P46063 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12130343 0.85 MGAM (0.56) ALDH1A1MAPTGAAMGAMHDAC8
SCHEMBL5158144 0.83 ALDH1A1 (0.57) ALDH1A1MAPTGAAMGAMHDAC8
SCHEMBL5160087 0.83 ALDH1A1 (0.58) ALDH1A1MAPTGAAMGAMHDAC8
SCHEMBL5163053 0.83 ALDH1A1 (0.70) ALDH1A1MAPTGAAMGAMHDAC8
SCHEMBL8237398 0.82 MGAM (0.61) ALDH1A1MAPTGAAMGAMHDAC8
SCHEMBL30417045 0.82 MGAM (0.61) ALDH1A1MAPTGAAMGAMHDAC8
SCHEMBL17035499 0.82 MAPT (0.64) ALDH1A1MAPTGAAMGAMHDAC8
SCHEMBL8906407 0.82 ALDH1A1 (0.55) ALDH1A1MAPTGAAMGAMHDAC8
SCHEMBL5161504 0.82 ALDH1A1 (0.55) ALDH1A1MAPTGAAMGAMHDAC8
SCHEMBL5158859 0.81 ALDH1A1 (0.54) ALDH1A1MAPTGAAMGAMHDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0210284-B1 1,3-DITHIOL-2-YLIDENE DERIVATIVES BANYU PHARMACEUTICAL CO., LTD. (JP) 1992-08-19 EP disclosed
US-5112820-A Vision defects STERLING DRUG INC. (US) 1992-05-12 US disclosed
US-5109135-A 2- or 3-aminomethyl-4-amino-3,4-dihydro-2H-1,4-benzoxazine intermediates STERLING DRUG INC. (US) 1992-04-28 US disclosed
US-5066803-A Chemical intermediates for analgesics STERLING DRUG INC. (US) 1991-11-19 US disclosed
WO-1990007505-A1 2- AND 3-AMINOMETHYL-6-ARYLCARBONYL-2,3-DIHYDROPYRROLO[1,2,3-de]-1,4-BENZOXAZINES STERLING DRUG INC. (US) 1990-07-12 WO disclosed
US-4939138-A 2- and 3-aminomethyl-6-arylcarbonyl-2,3-dihydropyrrolo(1,2,3-DE)-1,4-benzoxazines STERLING DRUG INC. (US) 1990-07-03 US disclosed
US-4668799-A Anti-hepatitis and anti-cirrhotic 1,3-dithiol-2-ylidene derivatives, and pharmaceutical compositions therefor BANYU PHARMACEUTICAL CO., LTD. (JP) 1987-05-26 US disclosed
EP-0210284-A1 1,3-Dithiol-2-ylidene derivatives BANYU PHARMACEUTICAL CO., LTD. (JP) 1987-02-04 EP disclosed