SCHEMBL9669141

SCHEMBL9669141

O=C1CNC(c2ccc3[nH]c(-c4cncnc4)cc3c2)=NN1

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CDK5 Q00535 5/20 0.39
CDK5R1 Q15078 5/20 0.39
CYP19A1 P11511 3/20 0.37
IDH1 O75874 1/20 0.32
CLK2 P49760 3/20 0.32
CLK3 P49761 3/20 0.32
DYRK1A Q13627 3/20 0.32
MAPKAPK2 P49137 1/20 0.32
NAMPT P43490 1/20 0.31
SYK P43405 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9669186 0.88 CDC7 (0.40) CDK5CDK5R1CYP19A1CLK2DYRK1A
SCHEMBL9667854 0.80 ABL1 (0.34) CDK5CDK5R1CYP19A1
SCHEMBL9669379 0.80 PDE3B (0.45) CDK5CDK5R1
SCHEMBL9669065 0.70 CYP19A1 (0.52) CDK5CDK5R1CYP19A1CLK2CLK3
SCHEMBL9669332 0.69 CDK5 (0.41) CDK5CDK5R1CYP19A1IDH1CLK2
SCHEMBL9667675 0.68 KCNH2 (0.52)
SCHEMBL9669307 0.67 MAOB (0.43)
SCHEMBL7355155 0.67 KCNH2 (0.44)
SCHEMBL22309145 0.67 PDE3B (0.42)
SCHEMBL4211464 0.67 PDE3B (0.51)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0223937-B1 INDOLES SUBSTITUTED WITH HETEROCYCLES, INTERMEDIATES, PROCESS FOR THEIR PREPARATION AND MEDICAMENTS Roche Diagnostics GmbH (DE) 1992-03-18 EP disclosed
US-4851406-A CARDIOVASCULAR DISORDERS, HYPOTENSIVE BOEHRINGER MANNHEIM GMBH (DE) 1989-07-25 US disclosed