SCHEMBL22309145

SCHEMBL22309145

O=C1CNC(c2ccc(F)c(F)c2)=NN1

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 10/20 0.42
PDE3A Q14432 10/20 0.42
NOTUM Q6P988 1/20 0.40
PGR P06401 1/20 0.36
NISCH Q9Y2I1 2/20 0.36
CYP17A1 P05093 1/20 0.35
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35
TRPA1 O75762 1/20 0.35
IDO1 P14902 1/20 0.34
KMO O15229 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4196668 0.88 PARP1 (0.43) PDE3BPDE3ANISCH
SCHEMBL22309155 0.84 PDE3B (0.47) PDE3BPDE3AKMO
SCHEMBL22308341 0.80 MAPT (0.39) PDE3BPDE3A
SCHEMBL4215079 0.78 MAOB (0.43) NOTUM
SCHEMBL22308892 0.78 PDE3B (0.62) PDE3BPDE3A
SCHEMBL22309151 0.78 PDE3B (0.48) PDE3BPDE3A
SCHEMBL4211464 0.77 PDE3B (0.51) PDE3BPDE3ANOTUMNISCHKMO
SCHEMBL10899939 0.76 PGR (0.42) NOTUMPGR
SCHEMBL22308851 0.75 PDE3B (0.54) PDE3BPDE3ANOTUM
SCHEMBL4215979 0.75 PDE3B (0.32) PDE3BPDE3APGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020157189-A1 1,2,4-TRIAZIN-6(1H)-ONE COMPOUNDS FOR THE TREATMENT OF HYPERPROLIFERATIVE DISEASES BAYER AKTIENGESELLSCHAFT (DE) 2020-08-06 WO disclosed