SCHEMBL9670429

SCHEMBL9670429

Oc1nc2ccc3c(Br)cccc3c2nc1O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TYMS P04818 2/20 0.41
BACE1 P56817 1/20 0.41
MYC P01106 1/20 0.40
MAX P61244 1/20 0.40
GUSB P08236 1/20 0.36
ACHE P22303 1/20 0.35
PLAU P00749 1/20 0.35
NQO2 P16083 2/20 0.33
PRNP P04156 1/20 0.33
CYP1A2 P05177 1/20 0.33
PARP1 P09874 1/20 0.33
GRM5 P41594 1/20 0.33
KCNH2 Q12809 1/20 0.33
KMT2A Q03164 3/20 0.32
GAA P10253 2/20 0.32
MAPT P10636 2/20 0.32
RAB9A P51151 2/20 0.32
ALDH1A1 P00352 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
CDK9 P50750 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9670911 0.84 MYC (0.49) MYCMAXNQO2PRNPCYP1A2
SCHEMBL5142239 0.76 CDK2 (0.56) MYCMAXACHECYP1A2KMT2A
SCHEMBL9670627 0.75 HTT (0.39) MYCMAXACHEKMT2AGAA
SCHEMBL9670672 0.73 TTR (0.47) MYCMAXCYP1A2KMT2AALDH1A1
SCHEMBL5886268 0.73 ALDH1A1 (0.58) TYMSBACE1PRNPKMT2AALDH1A1
SCHEMBL9578558 0.73 PRMT5 (0.49) MYCMAXCYP1A2RAB9AALDH1A1
SCHEMBL9671082 0.69 MYC (0.49) MYCMAXACHENQO2CYP1A2
SCHEMBL1248415 0.68 PARP1 (0.50) TYMSBACE1PLAUPRNPCYP1A2
SCHEMBL1489217 0.68 PARP1 (0.54) TYMSBACE1PLAUPRNPCYP1A2
SCHEMBL29375428 0.68 PARP1 (0.54) TYMSBACE1PLAUPRNPCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4889855-A ADMINISTERING GLUTAMATE ANTAGONIST TO INHIBIT HYPERACTIVITY OF EXCITATORY NEUROTRANSMITTERS A/S FERROSAN (DK) 1989-12-26 US claimed
EP-0283959-B1 HETEROCYCLIC COMPOUNDS AND THEIR PREPARATION AND USE NOVO NORDISK A/S (DK) 1992-01-02 EP disclosed
US-4912108-A Containing hydroxy substitution A/S FERROSAN (DK) 1990-03-27 US disclosed
US-4889855-A ADMINISTERING GLUTAMATE ANTAGONIST TO INHIBIT HYPERACTIVITY OF EXCITATORY NEUROTRANSMITTERS A/S FERROSAN (DK) 1989-12-26 US disclosed
EP-0283959-A1 Heterocyclic compounds and their preparation and use NOVO NORDISK A/S (DK) 1988-09-28 EP disclosed