SCHEMBL9674286

SCHEMBL9674286

CC(=O)N(N)c1ccc(O)c(O)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 8/20 0.48
HSD17B10 Q99714 6/20 0.48
RECQL P46063 5/20 0.48
HIF1A Q16665 5/20 0.48
TDP1 Q9NUW8 5/20 0.48
HPGD P15428 5/20 0.48
POLB P06746 4/20 0.48
ALOX15 P16050 4/20 0.48
ALDH1A1 P00352 4/20 0.48
BLM P54132 4/20 0.48
USP2 O75604 3/20 0.48
MEN1 O00255 3/20 0.48
APEX1 P27695 3/20 0.48
KMT2A Q03164 3/20 0.48
RGS12 O14924 2/20 0.48
THRB P10828 2/20 0.48
NFKB1 P19838 2/20 0.48
BRCA1 P38398 2/20 0.48
GNAI1 P63096 2/20 0.48
PKM P14618 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9673110 0.82 KDM4E (0.46) KDM4EHSD17B10RECQLHIF1ATDP1
SCHEMBL28157600 0.79 KDM4E (0.44) KDM4EHSD17B10RECQLHIF1ATDP1
SCHEMBL11800568 0.79 KDM4E (0.52) KDM4EHSD17B10RECQLHIF1ATDP1
SCHEMBL11793624 0.78 SMN1; SMN2 (0.55) KDM4EHSD17B10RECQLHIF1ATDP1
SCHEMBL5663915 0.77 ESR1 (0.41) KDM4EHSD17B10RECQLHIF1AHPGD
SCHEMBL4351797 0.76 ALDH1A1 (0.45) TDP1POLBALDH1A1SMN1; SMN2MAPT
SCHEMBL10441674 0.74 HDAC3 (0.40) HSD17B10MEN1APEX1KMT2ASMN1; SMN2
SCHEMBL31572011 0.74 TDP1 (0.55) KDM4EHSD17B10RECQLHIF1ATDP1
SCHEMBL6346993 0.73 SMN1; SMN2 (0.46) KDM4EHSD17B10RECQLHIF1ATDP1
SCHEMBL8502015 0.73 KDM4E (0.46) KDM4EHSD17B10RECQLHIF1ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0251143-B1 2-Oxo-1-[[(Substituted Sulfonyl)Amino]-Carbonyl]Azetidines Bristol-Myers Squibb GmbH (DE) 1992-08-26 EP disclosed
US-4801705-A 2-oxo-1-(((substituted sulfonyl)amino)-carbonyl)azetidines E. R. SQUIBB & SONS, INC. (US) 1989-01-31 US disclosed
EP-0251143-A1 2-Oxo-1-[[(Substituted Sulfonyl)Amino]-Carbonyl]Azetidines Bristol-Myers Squibb GmbH (DE) 1988-01-07 EP disclosed