SCHEMBL967510

SCHEMBL967510

Cc1c(N)nc(N)c(N)c1C

nearest known ligand 0.36

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.36
PDE10A Q9Y233 1/20 0.32
NOS1 P29475 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11581915 0.87 LMNA (0.39) LMNAPDE10ANOS1
Hydrochloric Acid SCHEMBL11582940 0.84 LMNA (0.38) LMNANOS1
SCHEMBL3670530 0.83 LMNA (0.41) LMNAPDE10ANOS1
SCHEMBL20869795 0.80 LMNA (0.39) LMNAPDE10ANOS1
SCHEMBL2067816 0.79 LMNA (0.46) LMNAPDE10ANOS1
SCHEMBL2284408 0.79 LMNA (0.46) LMNANOS1
Hydrochloric Acid SCHEMBL4932899 0.77 LMNA (0.44) LMNAPDE10A
SCHEMBL5924277 0.73 LMNA (0.46) LMNANOS1
SCHEMBL28173266 0.69 HSP90AA1 (0.32) LMNA
SCHEMBL8003108 0.69 HSP90AB1 (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110003866-A1 NOVEL 2-DIMETHYLAMINO-3-AMIDO-6-AMINO-PYRIDINE DERIVATIVES USEFUL AS POTASSIUM CHANNEL ACTIVATORS NEUROSEARCH A/S (DK) 2011-01-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110003866-A1 NOVEL 2-DIMETHYLAMINO-3-AMIDO-6-AMINO-PYRIDINE DERIVATIVES USEFUL AS POTASSIUM CHANNEL ACTIVATORS KCNA7, KCNJ2, KCNN3 LMNA 1847/4885PDE10A 869/4885NOS1 2771/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.