SCHEMBL9675810

SCHEMBL9675810

CC(=O)OCc1nc2cc(F)ccc2[nH]1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.45
SMN1; SMN2 Q16637 4/20 0.45
MAPK1 P28482 1/20 0.45
MEN1 O00255 1/20 0.43
LMNA P02545 1/20 0.43
KMT2A Q03164 1/20 0.43
HSD17B10 Q99714 3/20 0.41
ALDH1A1 P00352 3/20 0.41
KDM4E B2RXH2 2/20 0.41
MAOA P21397 2/20 0.40
MAOB P27338 2/20 0.40
IDO1 P14902 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
TSHR P16473 1/20 0.39
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9675828 0.89 IDO1 (0.54) MAPTSMN1; SMN2MAPK1MEN1LMNA
SCHEMBL9673902 0.80 MAPT (0.63) MAPTSMN1; SMN2LMNAHSD17B10ALDH1A1
SCHEMBL9513404 0.77 TSHR (0.47) MAPTSMN1; SMN2LMNAHSD17B10ALDH1A1
SCHEMBL9847737 0.76 HSD17B10 (0.54) MAPTSMN1; SMN2LMNAHSD17B10ALDH1A1
SCHEMBL8417202 0.76 DDAH1 (0.58) MAPTMEN1LMNAKMT2AHSD17B10
SCHEMBL5774011 0.76 TDP1 (0.51) LMNAHSD17B10ALDH1A1KDM4EIDO1
SCHEMBL13351516 0.73 IDO1 (0.54) KMT2AALDH1A1KDM4EIDO1
SCHEMBL8071535 0.73 HRH4 (0.47) MAPTLMNAHSD17B10ALDH1A1KDM4E
SCHEMBL20867740 0.72 IDO1 (0.57) ALDH1A1KDM4EIDO1F10
SCHEMBL1083641 0.72 IDO1 (0.49) ALDH1A1KDM4EIDO1RAB9AF10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0276942-B1 6-BETA(SUBSTITUTED)-(S)-HYDROXYMETHYLPENICILLANIC ACIDS AND DERIVATIVES THEREOF PFIZER INC. (US) 1992-04-01 EP disclosed
US-4782050-A BACTERICIDES PFIZER INC. (US) 1988-11-01 US disclosed
EP-0276942-A1 6-Beta(substituted)-(S)-hydroxymethylpenicillanic acids and derivatives thereof PFIZER INC. (US) 1988-08-03 EP disclosed