SCHEMBL9680324

SCHEMBL9680324

COc1cc2c(nc1C=O)CCC2

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.51
FGFR4 P22455 1/20 0.39
KDM4E B2RXH2 5/20 0.37
CYP19A1 P11511 2/20 0.37
CYP11B2 P19099 1/20 0.37
PDE4D Q08499 3/20 0.36
KMT2A Q03164 2/20 0.36
HSD17B10 Q99714 1/20 0.36
MEN1 O00255 1/20 0.35
MAPT P10636 2/20 0.34
CYP3A4 P08684 1/20 0.34
ALDH1A1 P00352 2/20 0.34
TSHR P16473 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
PRNP P04156 1/20 0.34
RXFP1 Q9HBX9 1/20 0.34
MAOB P27338 1/20 0.34
CDK5 Q00535 1/20 0.34
CDK5R1 Q15078 1/20 0.34
TUBB4A P04350 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9681811 0.74 NPC1 (0.44) NPC1KDM4EKMT2AHSD17B10MEN1
SCHEMBL28308539 0.73 PRNP (0.45) NPC1KDM4EHSD17B10MAPTALDH1A1
SCHEMBL5117887 0.73 NPC1 (0.53) NPC1KDM4EKMT2AHSD17B10MEN1
SCHEMBL9455514 0.71 KDM4E (0.52) NPC1KDM4EHSD17B10MAPTALDH1A1
SCHEMBL9682063 0.71 NPC1 (0.41) NPC1KDM4EKMT2AMEN1MAPT
SCHEMBL6333760 0.70 ALDH1A1 (0.59) NPC1KDM4EPDE4DKMT2AMEN1
SCHEMBL5114888 0.70 NPC1 (0.50) NPC1KDM4EPDE4DKMT2AHSD17B10
SCHEMBL6074387 0.69 FGFR4 (0.40) FGFR4CYP19A1CYP11B2PDE4DKMT2A
Acetic Acid SCHEMBL5125173 0.68 KDM4E (0.46) NPC1KDM4EKMT2AHSD17B10MEN1
SCHEMBL5045112 0.68 MAPT (0.62) KDM4ECYP19A1CYP11B2PDE4DMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0481802-A1 Hydroxylated inhibitors of HIV reverse transcriptase MERCK & CO. INC. (US) 1992-04-22 EP disclosed