SCHEMBL9681811

SCHEMBL9681811

COc1nc2c(cc1C=O)CCC2

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.44
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
GRM1 Q13255 2/20 0.36
KDM4E B2RXH2 6/20 0.35
ALDH1A1 P00352 6/20 0.35
TSHR P16473 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
PRNP P04156 1/20 0.34
RXFP1 Q9HBX9 1/20 0.34
MAPT P10636 6/20 0.34
SMN1; SMN2 Q16637 5/20 0.34
RAB9A P51151 4/20 0.34
LMNA P02545 2/20 0.34
CDK5 Q00535 1/20 0.34
CDK5R1 Q15078 1/20 0.34
TP53 P04637 1/20 0.34
MAPK1 P28482 1/20 0.34
HTT P42858 1/20 0.34
NFKB1 P19838 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9682063 0.97 NPC1 (0.41) NPC1MEN1KMT2AGRM1KDM4E
SCHEMBL7910316 0.75 SLC9A1 (0.49) NPC1MEN1KMT2AGRM1KDM4E
SCHEMBL9680324 0.74 NPC1 (0.51) NPC1MEN1KMT2AGRM1KDM4E
SCHEMBL25279182 0.73 POLB (0.45) NPC1MEN1KMT2AGRM1KDM4E
SCHEMBL30825541 0.71 KDM4E (0.59) NPC1MEN1KMT2AKDM4EALDH1A1
SCHEMBL6333760 0.70 ALDH1A1 (0.59) NPC1MEN1KMT2AKDM4EALDH1A1
SCHEMBL25274599 0.70 KDM4E (0.48) NPC1KMT2AGRM1KDM4EALDH1A1
SCHEMBL29580781 0.69 TDP1 (0.41) MEN1KMT2AKDM4EALDH1A1TSHR
SCHEMBL20539389 0.69 TDP1 (0.41) MEN1KMT2AKDM4EALDH1A1TSHR
SCHEMBL6073463 0.69 CYP11B1 (0.36) NPC1KDM4EALDH1A1TSHRTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0481802-A1 Hydroxylated inhibitors of HIV reverse transcriptase MERCK & CO. INC. (US) 1992-04-22 EP disclosed