SCHEMBL9680378

SCHEMBL9680378

Clc1ccccc1-n1nc(N2CCNCC2)c2ccccc21

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 2/20 0.58
CYP1A2 P05177 4/20 0.47
CYP2D6 P10635 3/20 0.47
CYP3A4 P08684 3/20 0.47
HSD17B10 Q99714 2/20 0.47
MAPT P10636 2/20 0.47
CYP2C19 P33261 2/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
DRD2 P14416 1/20 0.47
DRD3 P35462 1/20 0.47
HTR1A P08908 3/20 0.43
HTR6 P50406 2/20 0.43
HTR7 P34969 2/20 0.43
HTR3A P46098 2/20 0.43
HTR3E A5X5Y0 1/20 0.43
HTR3B O95264 1/20 0.43
NCF1 P14598 1/20 0.43
TSHR P16473 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9681936 0.99 ADRB1 (0.56) ADRB1CYP1A2CYP2D6CYP3A4HSD17B10
SCHEMBL9682493 0.85 ADRB1 (0.50) ADRB1CYP1A2CYP2D6CYP3A4HSD17B10
SCHEMBL9681356 0.84 DRD2 (0.47) CYP1A2CYP2D6CYP3A4HSD17B10MAPT
SCHEMBL9683176 0.84 SCN9A (0.48) CYP1A2CYP2D6HSD17B10MAPTHTR1A
Hydrochloric Acid SCHEMBL9683227 0.83 DRD2 (0.46) CYP1A2CYP2D6CYP3A4HSD17B10MAPT
Hydrochloric Acid SCHEMBL9681905 0.83 SCN9A (0.47) CYP1A2CYP2D6HSD17B10MAPTHTR1A
SCHEMBL2710715 0.80 KHK (0.54) ADRB1MAPTHTR6HTR3AHTR3E
Hydrochloric Acid SCHEMBL9681346 0.79 KHK (0.53) ADRB1MAPTHTR6HTR3AHTR3E
SCHEMBL9680660 0.79 PTGER1 (0.43) MAPTMEN1KMT2ADRD2HTR1A
SCHEMBL9683217 0.77 SCN9A (0.42) MAPTHTR1AHTR6HTR7HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4999356-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1991-03-12 US claimed
US-5134236-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-07-28 US disclosed
US-4999356-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1991-03-12 US disclosed
EP-0302423-A2 1-Phenyl-3-(1-piperazinyl)-1h-indazoles, a process and intermediates for their preparation, and the use thereof as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-02-08 EP disclosed