SCHEMBL9680653

SCHEMBL9680653

Cc1ccc(-n2nc(N3CCN(C(N)=O)CC3)c3ccccc32)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGER1 P34995 2/20 0.43
MAPT P10636 2/20 0.43
SMO Q99835 1/20 0.42
AKT1 P31749 1/20 0.42
AKT2 P31751 1/20 0.42
AKT3 Q9Y243 1/20 0.42
KMT2A Q03164 5/20 0.42
SMN1; SMN2 Q16637 3/20 0.42
TSHR P16473 2/20 0.42
HSD17B10 Q99714 2/20 0.42
MEN1 O00255 3/20 0.42
POLB P06746 1/20 0.42
ADRB2 P07550 1/20 0.42
ALDH1A1 P00352 4/20 0.41
LMNA P02545 4/20 0.41
NPSR1 Q6W5P4 3/20 0.41
MAPK1 P28482 2/20 0.41
HPGD P15428 1/20 0.41
ALOX15 P16050 1/20 0.41
RXFP1 Q9HBX9 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9681935 0.90 PTGER1 (0.49) PTGER1MAPTSMOKMT2ATSHR
SCHEMBL9763071 0.89 PTGER1 (0.44) PTGER1MAPTKMT2ASMN1; SMN2HSD17B10
SCHEMBL9680606 0.88 TP53 (0.45) PTGER1MAPTSMOAKT1AKT2
SCHEMBL9682459 0.87 POLB (0.47) MAPTSMOAKT1AKT2AKT3
SCHEMBL9763297 0.85 SCN9A (0.46) PTGER1MAPTAKT1AKT2AKT3
SCHEMBL16260557 0.83 MEN1 (0.53) MAPTKMT2ASMN1; SMN2MEN1POLB
SCHEMBL9762766 0.82 KHK (0.52) MAPTKMT2AMEN1HTTKHK
Hydrochloric Acid SCHEMBL9681492 0.81 KHK (0.51) MAPTKMT2AMEN1HTTKHK
SCHEMBL9681867 0.79 KHK (0.53) KHK
SCHEMBL9681280 0.79 LMNA (0.45) PTGER1MAPTKMT2ASMN1; SMN2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4999356-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1991-03-12 US claimed
US-5134236-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-07-28 US disclosed
US-4999356-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1991-03-12 US disclosed
EP-0302423-A2 1-Phenyl-3-(1-piperazinyl)-1h-indazoles, a process and intermediates for their preparation, and the use thereof as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-02-08 EP disclosed