SCHEMBL9681935

SCHEMBL9681935

NC(=O)N1CCN(c2nn(-c3ccccc3)c3ccccc23)CC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGER1 P34995 2/20 0.49
HTR1A P08908 1/20 0.45
HTR2A P28223 1/20 0.45
HTR7 P34969 1/20 0.45
HTR6 P50406 1/20 0.45
SCN9A Q15858 1/20 0.44
ALDH1A1 P00352 4/20 0.42
LMNA P02545 1/20 0.42
MAPT P10636 3/20 0.41
RAB9A P51151 1/20 0.41
TP53 P04637 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
KHK P50053 1/20 0.40
FAAH O00519 1/20 0.40
MGLL Q99685 1/20 0.40
SMO Q99835 1/20 0.40
KIT P10721 1/20 0.39
CDK1 P06493 1/20 0.39
IGF1R P08069 1/20 0.39
FGFR1 P11362 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9763071 0.91 PTGER1 (0.44) PTGER1HTR1AHTR2AHTR7HTR6
SCHEMBL9680653 0.90 PTGER1 (0.43) PTGER1SCN9AALDH1A1LMNAMAPT
SCHEMBL9680606 0.90 TP53 (0.45) PTGER1SCN9ALMNAMAPTTP53
SCHEMBL9682459 0.87 POLB (0.47) SCN9ALMNAMAPTTP53FAAH
SCHEMBL9763297 0.87 SCN9A (0.46) PTGER1SCN9ALMNAMAPTRAB9A
SCHEMBL9681937 0.86 KHK (0.42) PTGER1HTR1AHTR2AHTR7HTR6
SCHEMBL9680636 0.83 SMO (0.50) PTGER1ALDH1A1LMNAMAPTTP53
SCHEMBL9681280 0.83 LMNA (0.45) PTGER1SCN9AALDH1A1LMNAMAPT
SCHEMBL9680660 0.83 PTGER1 (0.43) PTGER1HTR1AHTR2AHTR7HTR6
SCHEMBL9681416 0.82 KMT2A (0.58) HTR1AALDH1A1LMNAMAPTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4999356-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1991-03-12 US claimed
US-5134236-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-07-28 US disclosed
US-4999356-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1991-03-12 US disclosed
EP-0302423-A2 1-Phenyl-3-(1-piperazinyl)-1h-indazoles, a process and intermediates for their preparation, and the use thereof as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-02-08 EP disclosed