SCHEMBL9680787

SCHEMBL9680787

Nc1cccc(C#Cc2ccc(SC(F)(F)F)cc2)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.52
ALDH1A1 P00352 1/20 0.52
TDP1 Q9NUW8 1/20 0.52
FFAR1 O14842 1/20 0.44
MAPT P10636 2/20 0.40
ADRB2 P07550 1/20 0.40
RAB9A P51151 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
PIK3CA P42336 1/20 0.38
MTOR P42345 1/20 0.38
PDK1 Q15118 1/20 0.38
HCRTR1 O43613 1/20 0.38
TSHR P16473 2/20 0.38
MAPK1 P28482 2/20 0.38
ASIC3 Q9UHC3 1/20 0.37
APP P05067 1/20 0.36
LMNA P02545 1/20 0.36
HTT P42858 1/20 0.36
PTPRZ1 P23471 2/20 0.36
CA12 O43570 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6001741 0.80 ALDH1A1 (0.56) KDM4EALDH1A1TDP1MAPTRAB9A
SCHEMBL9611202 0.80 FFAR1 (0.59) KDM4EALDH1A1TDP1FFAR1MAPT
SCHEMBL4970529 0.77 MAPT (0.67) FFAR1MAPTADRB2RAB9AL3MBTL1
SCHEMBL9611201 0.77 MAPT (0.67) FFAR1MAPTADRB2RAB9AL3MBTL1
SCHEMBL4968126 0.76 CYP3A4 (0.58) ALDH1A1TDP1FFAR1MAPTADRB2
SCHEMBL9195087 0.75 FFAR1 (0.51) FFAR1MAPTADRB2RAB9AL3MBTL1
SCHEMBL29574292 0.75 ALDH1A1 (0.56) KDM4EALDH1A1TDP1MAPTTSHR
SCHEMBL656796 0.75 ALDH1A1 (0.56) KDM4EALDH1A1TDP1MAPTTSHR
SCHEMBL29462452 0.74 MAPT (0.62) KDM4EALDH1A1TDP1FFAR1MAPT
SCHEMBL2811255 0.74 MAPT (0.62) KDM4EALDH1A1TDP1FFAR1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0493650-A1 Fluorinated acetylene-containing aromatic amines and diamines National Starch and Chemical Investment Holding Corporation (US) 1992-07-08 EP disclosed
US-5107026-A Fluorinated acetylene-containing aromatic amines and diamines NATIONAL STARCH AND CHEMICAL INVESTMENT HOLDING CORPORATION (US) 1992-04-21 US disclosed