SCHEMBL9680870

SCHEMBL9680870

CCc1cc(/C=C/c2cc(CC)c(COCc3ccccc3)[nH]c2=O)c(OC)nc1C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK5 Q00535 2/20 0.39
CDK5R1 Q15078 2/20 0.39
ALDH1A1 P00352 2/20 0.36
HCAR2 Q8TDS4 3/20 0.35
MMP13 P45452 1/20 0.34
PDE10A Q9Y233 3/20 0.34
GRM1 Q13255 1/20 0.33
TK1 P04183 1/20 0.32
PDE3B Q13370 1/20 0.31
PDE3A Q14432 1/20 0.31
ABL1 P00519 1/20 0.31
LCK P06239 1/20 0.31
LYN P07948 1/20 0.31
SRC P12931 1/20 0.31
CSK P41240 1/20 0.31
BTK Q06187 1/20 0.31
PTK6 Q13882 1/20 0.31
DHODH Q02127 1/20 0.31
MEN1 O00255 1/20 0.31
HSP90AA1 P07900 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9680874 1.00 CDK5 (0.39) CDK5CDK5R1ALDH1A1HCAR2MMP13
SCHEMBL9846195 0.78 PDE3B (0.36) ALDH1A1HCAR2PDE10APDE3BPDE3A
SCHEMBL9846194 0.78 PDE3B (0.36) ALDH1A1HCAR2PDE10APDE3BPDE3A
SCHEMBL9682778 0.74 HCAR2 (0.36) CDK5CDK5R1HCAR2
SCHEMBL9682775 0.74 HCAR2 (0.36) CDK5CDK5R1HCAR2
SCHEMBL9680279 0.70 TSHR (0.41) CDK5CDK5R1ALDH1A1HCAR2PDE10A
SCHEMBL9449305 0.68 SMN1; SMN2 (0.47) CDK5CDK5R1ALDH1A1HCAR2PDE3B
SCHEMBL9338308 0.67 L3MBTL1 (0.48) ALDH1A1HCAR2GRM1MEN1HSP90AA1
SCHEMBL9455953 0.67 TSHR (0.38) CDK5CDK5R1ALDH1A1HCAR2MEN1
Bromide SCHEMBL9682734 0.66 TSHR (0.37) CDK5CDK5R1ALDH1A1HCAR2MMP13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0481802-A1 Hydroxylated inhibitors of HIV reverse transcriptase MERCK & CO. INC. (US) 1992-04-22 EP disclosed